Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50012548
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558239BDBM50558239(CHEMBL4781228)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558245BDBM50558245(CHEMBL4789661)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558234BDBM50558234(CHEMBL4780536)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558243BDBM50558243(CHEMBL4746550)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558238BDBM50558238(CHEMBL4741579)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558241BDBM50558241(CHEMBL4760149)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558235BDBM50558235(CHEMBL4799043)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558247BDBM50558247(CHEMBL4749344)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558248BDBM50558248(CHEMBL4751840)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558242BDBM50558242(CHEMBL4799839)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558246BDBM50558246(CHEMBL4795251)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558240BDBM50558240(CHEMBL4786794)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558236BDBM50558236(CHEMBL4793078)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558237BDBM50558237(CHEMBL4788022)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558249BDBM50558249(CHEMBL4748287)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558244BDBM50558244(CHEMBL4751353)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558235BDBM50558235(CHEMBL4799043)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558237BDBM50558237(CHEMBL4788022)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558236BDBM50558236(CHEMBL4793078)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558234BDBM50558234(CHEMBL4780536)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]+/-DOI from human recombinant 5-HT2C receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558234BDBM50558234(CHEMBL4780536)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558234BDBM50558234(CHEMBL4780536)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ketanserin human recombinant 5-HT2A receptor after 60 mins by scintillation counting analysis relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Normandie Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558238BDBM50558238(CHEMBL4741579)
Affinity DataKi:  834nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed