TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 2.60E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University
Curated by ChEMBL
Kazan (Volga Region) Federal University
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair