Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50009851
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532879(CHEMBL3347611)
Affinity DataIC50: 27nMAssay Description:Inhibition of full-length GST-tagged CARM1 (unknown origin) using histone H3 substrate and [3H]SAM by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532879(CHEMBL3347611)
Affinity DataIC50: 27nMAssay Description:Inhibition of full-length GST-tagged CARM1 (unknown origin) using histone H3 substrate and [3H]SAM by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50158100(CHEMBL1614812)
Affinity DataIC50: 30nMAssay Description:Inhibition of full-length GST-tagged CARM1 (unknown origin) using histone H3 substrate and [3H]SAM by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50158100(CHEMBL1614812)
Affinity DataIC50: 30nMAssay Description:Inhibition of full-length GST-tagged CARM1 (unknown origin) using histone H3 substrate and [3H]SAM by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 50nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 50nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532877(CHEMBL4458225)
Affinity DataIC50: 220nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532877(CHEMBL4458225)
Affinity DataIC50: 220nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532858(CHEMBL4438506)
Affinity DataIC50: 240nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532858(CHEMBL4438506)
Affinity DataIC50: 240nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532867(CHEMBL4518126)
Affinity DataIC50: 270nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532867(CHEMBL4518126)
Affinity DataIC50: 270nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532876(CHEMBL4576510)
Affinity DataIC50: 360nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532876(CHEMBL4576510)
Affinity DataIC50: 360nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532869(CHEMBL4519457)
Affinity DataIC50: 400nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532869(CHEMBL4519457)
Affinity DataIC50: 400nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532868(CHEMBL4469882)
Affinity DataIC50: 410nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532868(CHEMBL4469882)
Affinity DataIC50: 410nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532869(CHEMBL4519457)
Affinity DataIC50: 600nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532866(CHEMBL4475924)
Affinity DataIC50: 600nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532869(CHEMBL4519457)
Affinity DataIC50: 600nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532866(CHEMBL4475924)
Affinity DataIC50: 600nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532868(CHEMBL4469882)
Affinity DataIC50: 700nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532868(CHEMBL4469882)
Affinity DataIC50: 700nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532877(CHEMBL4458225)
Affinity DataIC50: 800nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532877(CHEMBL4458225)
Affinity DataIC50: 800nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532858(CHEMBL4438506)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532858(CHEMBL4438506)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532870(CHEMBL4472656)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532870(CHEMBL4472656)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532861(CHEMBL4465484)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532860(CHEMBL4445795)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532860(CHEMBL4445795)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532861(CHEMBL4465484)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532862(CHEMBL4461242)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532862(CHEMBL4461242)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532860(CHEMBL4445795)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532860(CHEMBL4445795)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532876(CHEMBL4576510)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532876(CHEMBL4576510)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532870(CHEMBL4472656)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532870(CHEMBL4472656)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of PRMT6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of PRMT8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of PRMT8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532871(CHEMBL4470484)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of full-length Halo-tagged human CARM1 (1 to 608 residues) expressed in 293-F cells using [3H]-SAM and biotinylated histone peptides by sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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