Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50010219
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536316BDBM50536316(CHEMBL4537058)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536316BDBM50536316(CHEMBL4537058)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536333BDBM50536333(CHEMBL4550547)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536313BDBM50536313(CHEMBL4529072)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536342BDBM50536342(CHEMBL4548193)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536358BDBM50536358(CHEMBL2164269)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536348BDBM50536348(CHEMBL4545777)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536319BDBM50536319(CHEMBL4566039)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536344BDBM50536344(CHEMBL600947 | GNF-Pf-2911)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536329BDBM50536329(CHEMBL1995377)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536340BDBM50536340(CHEMBL4528019)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 42286BDBM42286(MLS000034309 | cid_654122 | N*2*-(2,5-Dimethoxy-ph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536311BDBM50536311(CHEMBL4593946)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536325BDBM50536325(CHEMBL4483432)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536338BDBM50536338(CHEMBL4542920)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536335BDBM50536335(CHEMBL4563650)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536321BDBM50536321(CHEMBL1622765)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536320BDBM50536320(CHEMBL4590509)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536326BDBM50536326(CHEMBL4534844)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536323BDBM50536323(CHEMBL4080220)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536322BDBM50536322(CHEMBL604514 | GNF-Pf-4167)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536324BDBM50536324(CHEMBL4072223)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536334BDBM50536334(CHEMBL3715362)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50402265BDBM50402265(CHEMBL2164280 | US8802861, 1)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536334BDBM50536334(CHEMBL3715362)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536361BDBM50536361(CHEMBL1613587)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536359BDBM50536359(CHEMBL4527282)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536312BDBM50536312(CHEMBL1458296)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536354BDBM50536354(CHEMBL1305300)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536352BDBM50536352(CHEMBL4561613)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536345BDBM50536345(CHEMBL4519027)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536314BDBM50536314(CHEMBL4543595)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536356BDBM50536356(CHEMBL4591485)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536318BDBM50536318(CHEMBL373492)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536343BDBM50536343(CHEMBL4581349)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536357BDBM50536357(CHEMBL4553536)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536341BDBM50536341(CHEMBL4520393)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536336BDBM50536336(CHEMBL4536891)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536327BDBM50536327(CHEMBL4526718)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536355BDBM50536355(CHEMBL4569913)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536346BDBM50536346(CHEMBL4544171)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536339BDBM50536339(CHEMBL4532396)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536351BDBM50536351(CHEMBL4567734)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536328BDBM50536328(CHEMBL1448756)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536362BDBM50536362(CHEMBL4517346)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536337BDBM50536337(CHEMBL4559250)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536331BDBM50536331(CHEMBL4553877)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536315BDBM50536315(CHEMBL4556925)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536349BDBM50536349(CHEMBL1700355)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50536317BDBM50536317(CHEMBL4585396)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
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