Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50010227
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 75.9nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 102nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 102nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 166nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 166nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 182nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 182nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 195nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 195nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 254nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 295nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 331nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 331nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 355nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 355nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 372nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 479nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 479nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 479nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 479nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 537nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Positive allosteric modulation activity at rat M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acetyl ...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Human)
Vanderbilt University School of Medicine
Curated by ChEMBL
Vanderbilt University School of Medicine
Curated by ChEMBL
Affinity DataEC50: 562nMAssay Description:Positive allosteric modulation activity at human M4 receptor expressed in CHO cells co-expressing Gqi5 protein assessed as potentiation of EC20 acety...More data for this Ligand-Target Pair














