BindingDB PrimarySearch

Report error Found 422 Enz. Inhib. hit(s) with all data for entry = 50010235

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

IC50: <0.25nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Tyrosine-protein kinase BTK(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged BTK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Testis-specific serine/threonine-protein kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged STK22D expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase TBK1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human GST-tagged TBK1 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: 1nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536677(CHEMBL4532781)

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Ribosomal protein S6 kinase alpha-3(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged RPS6KA3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536692(CHEMBL4550486)

IC50: 1.30nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Tyrosine-protein kinase ABL1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.30nMAssay Description:Inhibition of full-length human His-tagged ABL1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Receptor-type tyrosine-protein kinase FLT3(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.90nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic FLT3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Death-associated protein kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.90nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 4(Mouse)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2nMAssay Description:Inhibition of MARK4 in mouse cortical neurons assessed as inhibition of okadaic acid-induced tau phosphorylation at S262 residue preincubated for 15 ...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536685(CHEMBL4528550)

IC50: 2nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Cyclin-dependent kinase 2(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.20nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase Chk1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.20nMAssay Description:Inhibition of full-length recombinant human His-tagged CHEK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536693(CHEMBL4552799)

IC50: 2.40nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Tyrosine-protein kinase HCK(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.80nMAssay Description:Inhibition of full-length human N-terminal GST-tagged HCK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Ephrin type-B receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.90nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic EPHB2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Ephrin type-A receptor 8(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.90nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic EPHA8 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536686(CHEMBL4562217)

IC50: 3nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Proto-oncogene tyrosine-protein kinase Src(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3nMAssay Description:Inhibition of full-length recombinant human His-tagged SRC expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Leucine-rich repeat serine/threonine-protein kinase 2(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.10nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.20nMAssay Description:Inhibition of full-length recombinant human GST-tagged DYRK1A expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Macrophage colony-stimulating factor 1 receptor(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.30nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic CSF1R expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Cytoplasmic tyrosine-protein kinase BMX(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.5nMAssay Description:Inhibition of full-length recombinant human His-tagged BMX expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Vascular endothelial growth factor receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.5nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic KDR expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Tyrosine-protein kinase Lck(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.90nMAssay Description:Inhibition of full-length recombinant human His-tagged LCK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Cyclin-dependent kinase 7(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.10nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK7 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

PC cid PC sid

Details Article PubMed

NUAK family SNF1-like kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.20nMAssay Description:Inhibition of full-length recombinant human His-tagged NUAK1 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Cyclin-dependent kinase 5 activator 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.40nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged CDK5/P25 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.60nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged AMPK alpha1/beta1/gamma1 expressed in baculovirus expression system by LanthaScreen as...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536681(CHEMBL4552628)

IC50: 5nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536676(CHEMBL4593028)

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Misshapen-like kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 6nMAssay Description:Inhibition of recombinant human His-tagged MINK1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

Details Article PubMed

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536678(CHEMBL4550702)

IC50: 6nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase 26(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 6.30nMAssay Description:Inhibition of full-length recombinant human GST-tagged MST4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Inhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 7.10nMAssay Description:Inhibition of full-length recombinant human GST-tagged IKK-epsilon expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Ribosomal protein S6 kinase beta-1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged RPS6KB1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536687(CHEMBL4579339)

IC50: 9nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Interleukin-1 receptor-associated kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 9nMAssay Description:Inhibition of recombinant human GST-tagged IRAK1 (194 to 712 residues) catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536689(CHEMBL4571737)

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536701(CHEMBL4543195)

IC50: 10nMAssay Description:Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate m...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged AMPK alpha1/beta1/gamma1 expressed in baculovirus expression system by LanthaScreen as...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Vascular endothelial growth factor receptor 2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic KDR expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase TBK1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST-tagged TBK1 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Cyclin-dependent kinase 5 activator 1(Human)
Merck And

Curated by ChEMBL

BDBM50536678(CHEMBL4550702)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged CDK5/P25 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

MAP/microtubule affinity-regulating kinase 3(Human)
Merck And

Curated by ChEMBL

BDBM50536680(CHEMBL4569165)

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase TBK1(Human)
Merck And

Curated by ChEMBL

BDBM50536678(CHEMBL4550702)

IC50: <10nMAssay Description:Inhibition of full-length recombinant human GST-tagged TBK1 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Dual specificity protein kinase CLK2(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged CLK2 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

Details Article PubMed

Death-associated protein kinase 1(Human)
Merck And

Curated by ChEMBL

BDBM50536675(CHEMBL4569508)

IC50: <10nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Displayed 1 to 50 (of 422 total ) | Next | Last >>

Filter my 422 hits

Targets 99▿
- MAP/microtubule affinity-regulating kinase 3 26
- Mitogen-activated protein kinase 8 8
- Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform 4
- 5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 4
- Tyrosine-protein kinase JAK1 4
- Receptor tyrosine-protein kinase erbB-2 4
- Hepatocyte growth factor receptor 4
- Non-receptor tyrosine-protein kinase TYK2 4
- Serine/threonine-protein kinase B-raf 4
- Glycogen synthase kinase-3 alpha 4
- Glycogen synthase kinase-3 beta 4
- Serine/threonine-protein kinase Nek6 4
- Protein kinase C iota type 4
- NUAK family SNF1-like kinase 1 4
- Receptor-type tyrosine-protein kinase FLT3 4
- Serine/threonine-protein kinase Nek4 4
- Serine/threonine-protein kinase Nek2 4
- Sphingosine kinase 1 4
- Serine/threonine-protein kinase PAK 1 4
- Protein kinase C theta type 4
- Tyrosine-protein kinase JAK3 4
- Dual specificity mitogen-activated protein kinase kinase 1 4
- MAP/microtubule affinity-regulating kinase 4 4
- Tyrosine-protein kinase JAK2 4
- Dual specificity mitogen-activated protein kinase kinase 6 4
- Tyrosine-protein kinase ZAP-70 4
- Leucine-rich repeat serine/threonine-protein kinase 2 4
- Serine/threonine-protein kinase Sgk1 4
- Ephrin type-A receptor 3 4
- Tyrosine-protein kinase BTK 4
- Tyrosine-protein kinase ITK/TSK 4
- Insulin-like growth factor 1 receptor 4
- Epidermal growth factor receptor 4
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 4
- Ribosomal protein S6 kinase beta-1 4
- RAF proto-oncogene serine/threonine-protein kinase 4
- Serine/threonine-protein kinase 26 4
- Cyclin-dependent kinase 2 4
- Ephrin type-B receptor 2 4
- MAP kinase-activated protein kinase 2 4
- Ephrin type-A receptor 8 4
- MAP kinase-activated protein kinase 5 4
- Death-associated protein kinase 1 4
- PAS domain-containing serine/threonine-protein kinase 4
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 4
- Beta-adrenergic receptor kinase 1 4
- Cyclin-dependent kinase 7 4
- Serine/threonine-protein kinase pim-1 4
- Serine/threonine-protein kinase TAO2 4
- Testis-specific serine/threonine-protein kinase 1 4
- Angiopoietin-1 receptor 4
- Mast/stem cell growth factor receptor Kit 4
- Serine/threonine-protein kinase MRCK alpha 4
- Protein-tyrosine kinase 6 4
- Mitogen-activated protein kinase 14 4
- Activin receptor type-1B 4
- Casein kinase II subunit alpha 4
- Cyclin-dependent kinase 5 activator 1 4
- Interleukin-1 receptor-associated kinase 4 4
- Cytoplasmic tyrosine-protein kinase BMX 4
- RAC-gamma serine/threonine-protein kinase 4
- Interleukin-1 receptor-associated kinase 1 4
- Tyrosine-protein kinase ABL1 4
- RAC-alpha serine/threonine-protein kinase 4
- Rho-associated protein kinase 2 4
- Rho-associated protein kinase 1 4
- Proto-oncogene tyrosine-protein kinase Src 4
- Mitogen-activated protein kinase 1 4
- 3-phosphoinositide-dependent protein kinase 1 4
- Tyrosine-protein kinase Lck 4
- NT-3 growth factor receptor 4
- Mitogen-activated protein kinase 9 4
- G protein-coupled receptor kinase 4 4
- Dual specificity protein kinase CLK2 4
- High affinity nerve growth factor receptor 4
- G protein-coupled receptor kinase 6 4
- Calcium/calmodulin-dependent protein kinase type IV 4
- Serine/threonine-protein kinase N1 4
- Tyrosine-protein kinase SYK 4
- Ribosomal protein S6 kinase alpha-3 4
- Serine/threonine-protein kinase TBK1 4
- Cyclin-T1/Cyclin-dependent kinase 9 4
- Aurora kinase B 4
- Vascular endothelial growth factor receptor 2 4
- Insulin receptor 4
- Tyrosine-protein kinase HCK 4
- Fibroblast growth factor receptor 2 4
- Serine/threonine-protein kinase PLK1 4
- Inhibitor of nuclear factor kappa-B kinase subunit beta 4
- Mitogen-activated protein kinase 13 4
- RAC-beta serine/threonine-protein kinase 4
- Casein kinase I isoform alpha 4
- Misshapen-like kinase 1 4
- Macrophage colony-stimulating factor 1 receptor 4
- cAMP-dependent protein kinase catalytic subunit alpha 4
- Protein kinase C zeta type 4
- Serine/threonine-protein kinase Chk2 4
- Serine/threonine-protein kinase Chk1 4
- SRSF protein kinase 1 4
Publications 1▿
- Bioorg Med Chem Lett 26: 4362-6 (2016) 422
Institutions 1▿
- Merck And 422
Affinity: 0.25 to 1.0E+5 nM▿
- IC50 422
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 3