Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50010257
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536873(CHEMBL4574913)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536873(CHEMBL4574913)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536869(CHEMBL4575939)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536869(CHEMBL4575939)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536879(CHEMBL4560281)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536879(CHEMBL4560281)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536872(CHEMBL4556775)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536878(CHEMBL4514474)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536878(CHEMBL4514474)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536872(CHEMBL4556775)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536870(CHEMBL4563511)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536870(CHEMBL4563511)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536868(CHEMBL4592407)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536868(CHEMBL4592407)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536875(CHEMBL4536893)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536875(CHEMBL4536893)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536874(CHEMBL4526798)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536874(CHEMBL4526798)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536880(CHEMBL4568674)
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536880(CHEMBL4568674)
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536877(CHEMBL4564168)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536877(CHEMBL4564168)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536871(CHEMBL4546916)
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536871(CHEMBL4546916)
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536876(CHEMBL4547558)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Key Laboratory of Industrial Fermentation Microbiology (Tianjin University of Science & Technology)

Curated by ChEMBL
LigandPNGBDBM50536876(CHEMBL4547558)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed