Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50047833
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of hypotonicity-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of hypotonicity-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair