Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50049060
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396097(CHEMBL2170856)
Affinity DataIC50: 230nMAssay Description:Inhibition of telomerase activity in human MDA-MB-435 cell lysate measured after 24 hrs by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396097(CHEMBL2170856)
Affinity DataIC50: 230nMAssay Description:Inhibition of telomerase activity in human U2OS cell lysate measured after 24 hrs by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50157547(7,8,3',4'-tetrahydroxyflavone | 2-(3,4-dihydroxyph...)
Affinity DataIC50: 740nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233825(CHEMBL4081286)
Affinity DataIC50: 969nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233823(CHEMBL4097807)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of telomerase activity in human U2OS cell lysate measured after 24 hrs by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233823(CHEMBL4097807)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of telomerase activity in human MDA-MB-435 cell lysate measured after 24 hrs by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233826(CHEMBL4090090)
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233824(CHEMBL4070673)
Affinity DataIC50: 1.73E+3nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50126186(2-(3-Naphthalen-2-yl-but-2-enoylamino)-benzoic aci...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human telomerase activity isolated from HEK293 cells assessed as reduction in dNTP incorporation using 5'-biotinylated AATCCGTCGAGCAGAG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50126186(2-(3-Naphthalen-2-yl-but-2-enoylamino)-benzoic aci...)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233827(CHEMBL4076246)
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50233828(CHEMBL4062047)
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of telomerase activity (unknown origin) in cell free system using sulforhodamine labeled primer measured after 30 mins by telomerase repea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2019
Entry Details Article
PubMed