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Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 7441
TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195552(4-(((5-Mercapto-1,3,4-thiadiazol-2-yl)imino)methyl...)
Affinity DataIC50:  36nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195551(4-(((5-Mercapto-1,3,4-thiadiazol-2-yl)imino)methyl...)
Affinity DataIC50:  255nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195553(4-(((5-Mercapto-1,3,4-thiadiazol-2-yl)imino)methyl...)
Affinity DataIC50:  473nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195547(2-((2-Nitrobenzylidene)amino)-5-mercapto-1,3,4-thi...)
Affinity DataIC50:  671nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195548(2-((2-Methoxybenzylidene)amino)-5-mercapto-1,3,4-t...)
Affinity DataIC50:  733nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195540(2-((2-Fluorobenzylidene)amino)-5-mercapto-1,3,4-th...)
Affinity DataIC50:  765nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195550(2-(((5-Mercapto-1,3,4-thiadiazol-2-yl)imino)methyl...)
Affinity DataIC50:  785nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195554(2-((2,4,6-Trimethoxybenzylidene)amino)-5-mercapto-...)
Affinity DataIC50:  907nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195546(2-((4-(Tert-butyl)benzylidene)amino)-5-mercapto-1,...)
Affinity DataIC50:  1.39E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195544(4-Chloro-2-(((5-mercapto-1,3,4-thiadiazol-2-yl)imi...)
Affinity DataIC50:  1.72E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195545(4-Bromo-2-(((5-mercapto-1,3,4-thiadiazol-2-yl)imin...)
Affinity DataIC50:  1.97E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195542(2-((4-Chlorobenzylidene)amino)-5-mercapto-1,3,4-th...)
Affinity DataIC50:  2.46E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195543(2-((3,4-Dichlorobenzylidene)amino)-5-mercapto-1,3,...)
Affinity DataIC50:  3.62E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195541(2-((3-Chlorobenzylidene)amino)-5-mercapto-1,3,4-th...)
Affinity DataIC50:  4.75E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195549(2-((3,5-Dimethoxybenzylidene)amino)-5-mercapto-1,3...)
Affinity DataIC50:  5.35E+3nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  2.36E+4nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195539(2-(Benzylideneamino)-5-mercapto-1,3,4-thiadiazole ...)
Affinity DataIC50:  4.92E+4nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPolyphenol oxidase 1 [61-568](White button mushroom)
Shaoyang University

LigandPNGBDBM195555(2-(((5-(Benzylthio)-1,3,4-thiadiazol-2-yl)imino)me...)
Affinity DataIC50:  2.47E+5nMpH: 6.8Assay Description:Briefly, 1,3,4-thiadiazole derivatives were tested for diphenolase inhibitory activity of tyrosinase using L-DOPA (dihydroxyphenylalanine) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed