Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50009997
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534255BDBM50534255(CHEMBL4468662)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534253BDBM50534253(CHEMBL4579826)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534259BDBM50534259(CHEMBL4521500)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534251BDBM50534251(CHEMBL4449746)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534248BDBM50534248(CHEMBL4463440)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534254BDBM50534254(CHEMBL4543687)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534252BDBM50534252(CHEMBL4527984)
Affinity DataIC50: 17nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534261BDBM50534261(CHEMBL4443821)
Affinity DataIC50: 23nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203636BDBM50203636(CHEMBL3929715)
Affinity DataIC50: 44nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203630BDBM50203630(CHEMBL3891139)
Affinity DataIC50: 46nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534262BDBM50534262(CHEMBL4451197)
Affinity DataIC50: 62nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534244BDBM50534244(CHEMBL4556527)
Affinity DataIC50: 63nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534260BDBM50534260(CHEMBL4583030)
Affinity DataIC50: 64nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534249BDBM50534249(CHEMBL4522289)
Affinity DataIC50: 77nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534256BDBM50534256(CHEMBL4569903)
Affinity DataIC50: 103nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534247BDBM50534247(CHEMBL4519014)
Affinity DataIC50: 128nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534250BDBM50534250(CHEMBL4472601)
Affinity DataIC50: 167nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534241BDBM50534241(CHEMBL4557360)
Affinity DataIC50: 220nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203633BDBM50203633(CHEMBL3961252)
Affinity DataIC50: 248nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203552BDBM50203552(CHEMBL3943352)
Affinity DataIC50: 356nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534242BDBM50534242(CHEMBL4559431)
Affinity DataIC50: 462nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534245BDBM50534245(CHEMBL4472277)
Affinity DataIC50: 994nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203639BDBM50203639(CHEMBL3951486)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203629BDBM50203629(CHEMBL3911190)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534257BDBM50534257(CHEMBL4442898)
Affinity DataIC50: 3.76E+3nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534258BDBM50534258(CHEMBL4449662)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534243BDBM50534243(CHEMBL4459306)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sejong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534246BDBM50534246(CHEMBL4436175)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged full length human recombinant GSK3beta using [YRRAAVPPSPSLSRHSSPHQ-(pS)EDEEE] substrate and pre-incubarted for 20 mins befor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed