Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50010001
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393252BDBM50393252(CHEMBL2151570)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]A-585539 from alpha7 nAChR in human cerebral cortex membranes after 75 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 92878BDBM92878(Quinuclidine analogue, 5)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]MLA from alpha7 nAChR in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534298BDBM50534298(CHEMBL4438684)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534286BDBM50534286(CHEMBL4453542)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534287BDBM50534287(CHEMBL4519018)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to alpha3beta4 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500410BDBM50500410(CHEMBL3745799)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534288BDBM50534288(CHEMBL4472617)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534291BDBM50534291(CHEMBL4559236)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534294BDBM50534294(CHEMBL4460057)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]MLA from alpha7 nAChR in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534299BDBM50534299(CHEMBL4450133)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534300BDBM50534300(CHEMBL4442125)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534284BDBM50534284(CHEMBL4468804)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534292BDBM50534292(CHEMBL4437323)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534288BDBM50534288(CHEMBL4472617)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534289BDBM50534289(CHEMBL4535466)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534297BDBM50534297(CHEMBL4443082)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534296BDBM50534296(CHEMBL4557590)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534283BDBM50534283(CHEMBL4440403)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534282BDBM50534282(CHEMBL4437189)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534293BDBM50534293(CHEMBL3341966)
Affinity DataKi:  21nMAssay Description:Displacement of [3H] epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534293BDBM50534293(CHEMBL3341966)
Affinity DataKi:  21nMAssay Description:Displacement of [3H] epibatidine from alpha4beta2 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534302BDBM50534302(CHEMBL4463888)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534286BDBM50534286(CHEMBL4453542)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534295BDBM50534295(CHEMBL4521227)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534301BDBM50534301(CHEMBL4474896)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534285BDBM50534285(CHEMBL4453215)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534290BDBM50534290(CHEMBL4468230)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534292BDBM50534292(CHEMBL4437323)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500408BDBM50500408(CHEMBL3747760)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534297BDBM50534297(CHEMBL4443082)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534285BDBM50534285(CHEMBL4453215)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534288BDBM50534288(CHEMBL4472617)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]MLA from human recombinant alpha7 nAChR expressed in HEKtsA201 cells after 1 hr by CNiFERs binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534284BDBM50534284(CHEMBL4468804)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534283BDBM50534283(CHEMBL4440403)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534282BDBM50534282(CHEMBL4437189)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500409BDBM50500409(CHEMBL3747258)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534296BDBM50534296(CHEMBL4557590)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534291BDBM50534291(CHEMBL4559236)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534289BDBM50534289(CHEMBL4535466)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534300BDBM50534300(CHEMBL4442125)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500410BDBM50500410(CHEMBL3745799)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534287BDBM50534287(CHEMBL4519018)
Affinity DataKi:  221nMAssay Description:Binding affinity to alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534299BDBM50534299(CHEMBL4450133)
Affinity DataKi:  279nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534293BDBM50534293(CHEMBL3341966)
Affinity DataKi: >300nMAssay Description:Displacement of [3H] epibatidine from alpha7 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500409BDBM50500409(CHEMBL3747258)
Affinity DataKi:  362nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534299BDBM50534299(CHEMBL4450133)
Affinity DataKi:  414nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534292BDBM50534292(CHEMBL4437323)
Affinity DataKi:  449nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534286BDBM50534286(CHEMBL4453542)
Affinity DataKi:  461nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534287BDBM50534287(CHEMBL4519018)
Affinity DataKi:  476nMAssay Description:Binding affinity to alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Mahidol University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500410BDBM50500410(CHEMBL3745799)
Affinity DataKi:  515nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 76 total ) | Next | Last >>
Jump to: