Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50022531
TargetEpithelial discoidin domain-containing receptor 1(Human)
University Hospital and University of Zurich
Curated by ChEMBL
University Hospital and University of Zurich
Curated by ChEMBL
Affinity DataKd: 0.400nMAssay Description:Binding affinity to DDR1 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor Tie-1(Human)
University Hospital and University of Zurich
Curated by ChEMBL
University Hospital and University of Zurich
Curated by ChEMBL
Affinity DataKd: 0.900nMAssay Description:Binding affinity to TIE1 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
University Hospital and University of Zurich
Curated by ChEMBL
University Hospital and University of Zurich
Curated by ChEMBL
Affinity DataKd: 1.30nMAssay Description:Binding affinity to DDR2 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Inhibition of TIE2 autophosphorylation in human HUVEC cells by Western blot analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding affinity to TIE2 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 10(Human)
University Hospital and University of Zurich
Curated by ChEMBL
University Hospital and University of Zurich
Curated by ChEMBL
Affinity DataKd: 5.90nMAssay Description:Binding affinity to LOK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
