Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50048130
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205634(CHEMBL3933203)
Affinity DataIC50: 27nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205628(CHEMBL3906288)
Affinity DataIC50: 88nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205630(CHEMBL3915266)
Affinity DataIC50: 237nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205635(CHEMBL3898133)
Affinity DataIC50: 378nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205635(CHEMBL3898133)
Affinity DataIC50: 378nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205636(CHEMBL3923183)
Affinity DataIC50: 448nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205636(CHEMBL3923183)
Affinity DataIC50: 448nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205627(CHEMBL3914517)
Affinity DataIC50: 540nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205627(CHEMBL3914517)
Affinity DataIC50: 540nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205640(CHEMBL3901407)
Affinity DataIC50: 571nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205632(CHEMBL3901570)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205632(CHEMBL3901570)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205635(CHEMBL3898133)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205627(CHEMBL3914517)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205632(CHEMBL3901570)
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205626(CHEMBL3900506)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205626(CHEMBL3900506)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205626(CHEMBL3900506)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205633(CHEMBL3909213)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205633(CHEMBL3909213)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205636(CHEMBL3923183)
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205629(CHEMBL3905192)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205639(CHEMBL3892623)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205629(CHEMBL3905192)
Affinity DataIC50: 4.14E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205629(CHEMBL3905192)
Affinity DataIC50: 4.14E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205634(CHEMBL3933203)
Affinity DataIC50: 4.44E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205639(CHEMBL3892623)
Affinity DataIC50: 6.98E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205639(CHEMBL3892623)
Affinity DataIC50: 6.98E+3nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205628(CHEMBL3906288)
Affinity DataIC50: 7.75E+3nMAssay Description:Inhibition of human EZH1 complex using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205637(CHEMBL3896239)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205637(CHEMBL3896239)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205638(CHEMBL3929353)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205631(CHEMBL3975514)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205628(CHEMBL3906288)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Integral Biosciences

Curated by ChEMBL
LigandPNGBDBM50205634(CHEMBL3933203)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human wild type EZH2 using histone H3 as substrate after 1 hr in presence of 3H-SAM by filter paper detection analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2018
Entry Details Article
PubMed