Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50048928
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229700BDBM50229700(CHEMBL4085167)
Affinity DataEC50:  12nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229025BDBM50229025(CHEMBL4092421)
Affinity DataIC50: 13nMAssay Description:Inhibition of RIP1 (unknown origin) using MBP as substrate preincubated for 15 mins followed by MBP/ATP mixture addition measured after 90 mins by AD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Mouse)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229025BDBM50229025(CHEMBL4092421)
Affinity DataEC50:  27nMAssay Description:Inhibition of RIP1 in mouse L929 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 6 hrs by Cell Titer-Glo luminescent cell vi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229025BDBM50229025(CHEMBL4092421)
Affinity DataEC50:  28nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229585BDBM50229585(CHEMBL4076443)
Affinity DataEC50:  36nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228870BDBM50228870(CHEMBL4083065)
Affinity DataEC50:  49nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229606BDBM50229606(CHEMBL4072591)
Affinity DataEC50:  56nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229702BDBM50229702(CHEMBL4101314)
Affinity DataEC50:  58nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228873BDBM50228873(CHEMBL4063996)
Affinity DataEC50:  64nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229598BDBM50229598(CHEMBL4096278)
Affinity DataEC50:  72nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229605BDBM50229605(CHEMBL4061192)
Affinity DataEC50:  74nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229512BDBM50229512(CHEMBL4083937)
Affinity DataEC50:  98nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229699BDBM50229699(CHEMBL4059584)
Affinity DataEC50:  125nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228872BDBM50228872(CHEMBL4091760)
Affinity DataEC50:  198nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229541BDBM50229541(CHEMBL4096270)
Affinity DataEC50:  221nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228871BDBM50228871(CHEMBL4099502)
Affinity DataEC50:  262nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229517BDBM50229517(CHEMBL4068805)
Affinity DataEC50:  378nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229601BDBM50229601(CHEMBL4082828)
Affinity DataEC50:  457nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229242BDBM50229242(CHEMBL4084908)
Affinity DataEC50:  490nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229586BDBM50229586(CHEMBL4087013)
Affinity DataEC50:  627nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229515BDBM50229515(CHEMBL4076266)
Affinity DataEC50:  628nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229701BDBM50229701(CHEMBL4078224)
Affinity DataEC50:  628nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229429BDBM50229429(CHEMBL4092663)
Affinity DataEC50:  656nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36371BDBM36371(CID2828334 | 5-(1H-indol-3-ylmethyl)-3-methyl-2-th...)
Affinity DataIC50: 760nMAssay Description:Inhibition of recombinant GST-tagged RIP1 (unknown origin) after 4 hrs by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229587BDBM50229587(CHEMBL4080685)
Affinity DataEC50:  815nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229603BDBM50229603(CHEMBL4090332)
Affinity DataEC50:  898nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229028BDBM50229028(CHEMBL4066793)
Affinity DataEC50:  1.08E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229597BDBM50229597(CHEMBL4104038)
Affinity DataEC50:  1.23E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229422BDBM50229422(CHEMBL4102856)
Affinity DataEC50:  1.23E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229583BDBM50229583(CHEMBL4063537)
Affinity DataEC50:  1.25E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229610BDBM50229610(CHEMBL4073983)
Affinity DataEC50:  1.31E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229609BDBM50229609(CHEMBL4103563)
Affinity DataEC50:  1.53E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229552BDBM50229552(CHEMBL4095647)
Affinity DataEC50:  1.74E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229518BDBM50229518(CHEMBL4095053)
Affinity DataEC50:  2.53E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229188BDBM50229188(CHEMBL4096996)
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229510BDBM50229510(CHEMBL4073564)
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229187BDBM50229187(CHEMBL4085631)
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229588BDBM50229588(CHEMBL4086116)
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229228BDBM50229228(CHEMBL4069797)
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229025BDBM50229025(CHEMBL4092421)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229604BDBM50229604(CHEMBL4069288)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229026BDBM50229026(CHEMBL4095808)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229508BDBM50229508(CHEMBL4064968)
Affinity DataEC50:  8.24E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229703BDBM50229703(CHEMBL4080015)
Affinity DataEC50:  8.56E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229602BDBM50229602(CHEMBL4098042)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229582BDBM50229582(CHEMBL4086110)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229607BDBM50229607(CHEMBL4071625)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229513BDBM50229513(CHEMBL4092903)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229608BDBM50229608(CHEMBL4088080)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229509BDBM50229509(CHEMBL4100395)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
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