Compile Data Set for Download or QSAR
Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 50048942
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230401(CHEMBL4088079)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230385(CHEMBL4103682)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230386(CHEMBL4059902)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230398(CHEMBL4093905)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230369(CHEMBL4079379)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230372(CHEMBL4080203)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230411(SLV-319 | RAC-IBIPINABANT)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230406(CHEMBL4077774)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230370(CHEMBL4097409)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230414(CHEMBL4104443)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230377(CHEMBL4095928)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230379(CHEMBL4085754)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230381(CHEMBL4068564)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230383(CHEMBL4092420)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230408(CHEMBL4076361)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230370(CHEMBL4097409)
Affinity DataIC50: 18nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230403(CHEMBL4082778)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230383(CHEMBL4092420)
Affinity DataIC50: 19nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230386(CHEMBL4059902)
Affinity DataIC50: 22nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 25nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230368(CHEMBL4089687)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230396(CHEMBL4089263)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230382(CHEMBL4098324)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230397(CHEMBL4095806)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230380(CHEMBL4091555)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230407(CHEMBL4070659)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230384(CHEMBL4066919)
Affinity DataIC50: 30nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230396(CHEMBL4089263)
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230409(CHEMBL4100767)
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230371(CHEMBL4071282)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230401(CHEMBL4088079)
Affinity DataIC50: 40nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230384(CHEMBL4066919)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230408(CHEMBL4076361)
Affinity DataIC50: 50nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230404(CHEMBL4081820)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230416(CHEMBL4081392)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230413(CHEMBL4085630)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230373(CHEMBL4071623)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230400(CHEMBL4103562)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230414(CHEMBL4104443)
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230406(CHEMBL4077774)
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230415(CHEMBL4105652)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230376(CHEMBL4088193)
Affinity DataIC50: 70nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230405(CHEMBL4068077)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230403(CHEMBL4082778)
Affinity DataIC50: 72nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230378(CHEMBL4077892)
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230411(SLV-319 | RAC-IBIPINABANT)
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230409(CHEMBL4100767)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230374(CHEMBL4080344)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50230377(CHEMBL4095928)
Affinity DataIC50: 90nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2019
Entry Details Article
PubMed
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