Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50048943
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230572BDBM50230572(CHEMBL4078431)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230570BDBM50230570(CHEMBL4080720)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230421BDBM50230421(CHEMBL4060320)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230571BDBM50230571(CHEMBL4069003)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230567BDBM50230567(CHEMBL4070053)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230419BDBM50230419(CHEMBL4084847)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230568BDBM50230568(CHEMBL4097795)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230569BDBM50230569(CHEMBL4087646)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230562BDBM50230562(CHEMBL4079768)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230420BDBM50230420(CHEMBL4090083)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230564BDBM50230564(CHEMBL4097245)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230417BDBM50230417(CHEMBL4077956)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230422BDBM50230422(CHEMBL4091626)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230563BDBM50230563(CHEMBL4104950)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230565BDBM50230565(CHEMBL4061382)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230561BDBM50230561(CHEMBL4105530)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 68nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230566BDBM50230566(CHEMBL4097216)
Affinity DataIC50: 75nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230420BDBM50230420(CHEMBL4090083)
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230421BDBM50230421(CHEMBL4060320)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230419BDBM50230419(CHEMBL4084847)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230562BDBM50230562(CHEMBL4079768)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230561BDBM50230561(CHEMBL4105530)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230567BDBM50230567(CHEMBL4070053)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230571BDBM50230571(CHEMBL4069003)
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230563BDBM50230563(CHEMBL4104950)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230417BDBM50230417(CHEMBL4077956)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230570BDBM50230570(CHEMBL4080720)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230566BDBM50230566(CHEMBL4097216)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230422BDBM50230422(CHEMBL4091626)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230569BDBM50230569(CHEMBL4087646)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230564BDBM50230564(CHEMBL4097245)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230568BDBM50230568(CHEMBL4097795)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230565BDBM50230565(CHEMBL4061382)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230572BDBM50230572(CHEMBL4078431)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant human His-tagged HER2 cytoplasmic domain (676 to 1255 residues) expressed in baculovirus expression system using Poly (Glu,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2019
Entry Details Article
PubMed