Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50048142
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206258BDBM50206258(CHEMBL3963469)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206241BDBM50206241(CHEMBL3901366)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206256BDBM50206256(CHEMBL3917985)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206258BDBM50206258(CHEMBL3963469)
Affinity DataEC50:  18nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206268BDBM50206268(CHEMBL3891441)
Affinity DataEC50:  31nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206264BDBM50206264(CHEMBL3957600)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206240BDBM50206240(CHEMBL3928422)
Affinity DataEC50:  40nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206245BDBM50206245(CHEMBL3907100)
Affinity DataEC50:  41nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206264BDBM50206264(CHEMBL3957600)
Affinity DataEC50:  41nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206248BDBM50206248(CHEMBL3897030)
Affinity DataEC50:  45nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206240BDBM50206240(CHEMBL3928422)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206266BDBM50206266(CHEMBL3937435)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206266BDBM50206266(CHEMBL3937435)
Affinity DataEC50:  63nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206254BDBM50206254(CHEMBL3946303)
Affinity DataEC50:  70nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206251BDBM50206251(CHEMBL3951684)
Affinity DataEC50:  91nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206260BDBM50206260(CHEMBL3961124)
Affinity DataEC50:  95nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206244BDBM50206244(CHEMBL3969845)
Affinity DataEC50:  100nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206253BDBM50206253(CHEMBL3891068)
Affinity DataEC50:  120nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206261BDBM50206261(CHEMBL3931382)
Affinity DataEC50:  140nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206249BDBM50206249(CHEMBL3900048)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206262BDBM50206262(CHEMBL3909099)
Affinity DataEC50:  180nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206262BDBM50206262(CHEMBL3909099)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206244BDBM50206244(CHEMBL3969845)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206242BDBM50206242(CHEMBL3980345)
Affinity DataEC50:  250nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206256BDBM50206256(CHEMBL3917985)
Affinity DataEC50:  260nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206250BDBM50206250(CHEMBL3905979)
Affinity DataEC50:  260nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206246BDBM50206246(CHEMBL3919130)
Affinity DataEC50:  300nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206247BDBM50206247(CHEMBL3910223)
Affinity DataEC50:  320nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206250BDBM50206250(CHEMBL3905979)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206255BDBM50206255(CHEMBL3900472)
Affinity DataEC50:  410nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206243BDBM50206243(CHEMBL3918431)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206255BDBM50206255(CHEMBL3900472)
Affinity DataIC50: 690nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206241BDBM50206241(CHEMBL3901366)
Affinity DataEC50:  940nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206252BDBM50206252(CHEMBL3928032)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206265BDBM50206265(CHEMBL3909084)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206242BDBM50206242(CHEMBL3980345)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206248BDBM50206248(CHEMBL3897030)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206263BDBM50206263(CHEMBL3909492)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206254BDBM50206254(CHEMBL3946303)
Affinity DataIC50: 4.20E+3nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206263BDBM50206263(CHEMBL3909492)
Affinity DataEC50:  4.20E+3nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206247BDBM50206247(CHEMBL3910223)
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206249BDBM50206249(CHEMBL3900048)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at alpha7 nACh receptor (unknown origin) expressed in HEK293 cells assessed as increase in Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206251BDBM50206251(CHEMBL3951684)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206261BDBM50206261(CHEMBL3931382)
Affinity DataIC50: 1.90E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206253BDBM50206253(CHEMBL3891068)
Affinity DataIC50: 2.80E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206260BDBM50206260(CHEMBL3961124)
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206248BDBM50206248(CHEMBL3897030)
Affinity DataIC50: 3.40E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206252BDBM50206252(CHEMBL3928032)
Affinity DataIC50: 6.10E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206245BDBM50206245(CHEMBL3907100)
Affinity DataIC50: 7.10E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206268BDBM50206268(CHEMBL3891441)
Affinity DataIC50: 8.60E+4nMAssay Description:Antagonist activity at 5-HT3A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of Ca2+ flux by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: