TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human TG2 by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair