Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50048994
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 109086BDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232186BDBM50232186(CHEMBL4092049)
Affinity DataKd:  4.95E+3nMAssay Description:Binding affinity to NT-647-NHS-labelled KGA (unknown origin) after 10 mins by microscale thermophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50400050BDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232186BDBM50232186(CHEMBL4092049)
Affinity DataIC50: 9.89E+3nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232181BDBM50232181(CHEMBL4100547)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232189BDBM50232189(CHEMBL4064324)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232185BDBM50232185(CHEMBL4073733)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232180BDBM50232180(CHEMBL4084095)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232187BDBM50232187(CHEMBL4075531)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant KGA (unknown origin) using glutamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed