Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50049031
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233271(CHEMBL4071073)
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233271(CHEMBL4071073)
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233269(CHEMBL4100590)
Affinity DataIC50: 50nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233266(CHEMBL4092854)
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233266(CHEMBL4092854)
Affinity DataIC50: 290nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233272(CHEMBL4064246)
Affinity DataIC50: 300nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233264(CHEMBL4085105)
Affinity DataIC50: 300nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233273(CHEMBL4064664)
Affinity DataIC50: 350nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233267(CHEMBL4084142)
Affinity DataIC50: 350nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233273(CHEMBL4064664)
Affinity DataIC50: 550nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233265(CHEMBL4065193)
Affinity DataIC50: 600nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM20608([3H]4-OHT | cid_449459 | CHEMBL489 | AFIMOXIFENE |...)
Affinity DataIC50: 600nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM20608([3H]4-OHT | cid_449459 | CHEMBL489 | AFIMOXIFENE |...)
Affinity DataIC50: 650nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233268(CHEMBL4073790)
Affinity DataIC50: 750nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233268(CHEMBL4073790)
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233272(CHEMBL4064246)
Affinity DataIC50: 1.10E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233270(CHEMBL4091901)
Affinity DataIC50: 2.25E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233270(CHEMBL4091901)
Affinity DataIC50: 2.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM22435(4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-hy...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233269(CHEMBL4100590)
Affinity DataIC50: 2.78E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233267(CHEMBL4084142)
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR2(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM22435(4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-hy...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233264(CHEMBL4085105)
Affinity DataIC50: 5.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetEstrogen-related receptor gamma(Human)
The Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50233265(CHEMBL4065193)
Affinity DataIC50: 6.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed