Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50048954
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231335BDBM50231335(CHEMBL4105090)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231336BDBM50231336(CHEMBL4080854)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231330BDBM50231330(CHEMBL4100604)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231335BDBM50231335(CHEMBL4105090)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of HIF-1alpha transcriptional activity in human MCF7 cells assessed as reduction in VEGF secretion after 24 hrs under hypoxic condition by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229998BDBM50229998(CHEMBL4079051)
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231327BDBM50231327(CHEMBL4084153)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231387BDBM50231387(CHEMBL4061538)
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230936BDBM50230936(CHEMBL4081643)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231337BDBM50231337(CHEMBL4081784)
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231333BDBM50231333(CHEMBL4097377)
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230973BDBM50230973(CHEMBL4071087)
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231334BDBM50231334(CHEMBL4070201)
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231332BDBM50231332(CHEMBL4067317)
Affinity DataIC50: 2.94E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231389BDBM50231389(CHEMBL3804969)
Affinity DataIC50: 2.99E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229712BDBM50229712(CHEMBL4093734)
Affinity DataIC50: 3.27E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231385BDBM50231385(CHEMBL4089660)
Affinity DataIC50: 3.41E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231331BDBM50231331(CHEMBL4088570)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231329BDBM50231329(CHEMBL4073802)
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230650BDBM50230650(CHEMBL4099642)
Affinity DataIC50: 3.66E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231328BDBM50231328(CHEMBL3805951)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231382BDBM50231382(CHEMBL4099803)
Affinity DataIC50: 4.54E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229611BDBM50229611(CHEMBL4073033)
Affinity DataIC50: 4.54E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230135BDBM50230135(CHEMBL3805275)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in human MCF7 cells after 24 hrs under hypoxic condition by HRE lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2019
Entry Details Article
PubMed