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Found 56 Enz. Inhib. hit(s) with all data for entry = 50000940
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265482(CHEMBL4071661)
Affinity DataKi:  83nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265482(CHEMBL4071661)
Affinity DataKi:  90nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265524(CHEMBL4072651)
Affinity DataKi:  151nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265524(CHEMBL4072651)
Affinity DataKi:  151nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265525(CHEMBL4092454)
Affinity DataKi:  155nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265525(CHEMBL4092454)
Affinity DataKi:  160nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265478(CHEMBL3484893)
Affinity DataKi:  229nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265482(CHEMBL4071661)
Affinity DataKi:  230nMAssay Description:Antagonist activity at KOR (unknown origin) expressed in HTLA cells assessed as inhibition of Sal A-induced beta-arrestin recruitment preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265478(CHEMBL3484893)
Affinity DataKi:  230nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265482(CHEMBL4071661)
Affinity DataKi:  234nMAssay Description:Antagonist activity at KOR (unknown origin) expressed in HTLA cells assessed as inhibition of Sal A-induced beta-arrestin recruitment preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265477(CHEMBL4084706)
Affinity DataKi:  347nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265477(CHEMBL4084706)
Affinity DataKi:  350nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265518(CHEMBL4078777)
Affinity DataKi:  363nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265518(CHEMBL4078777)
Affinity DataKi:  380nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265507(CHEMBL4066432)
Affinity DataKi:  500nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265507(CHEMBL4066432)
Affinity DataKi:  501nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265476(CHEMBL1701606)
Affinity DataKi:  513nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265476(CHEMBL1701606)
Affinity DataKi:  520nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265475(CHEMBL4104275)
Affinity DataKi:  562nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265475(CHEMBL4104275)
Affinity DataKi:  562nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265458(CHEMBL4077345)
Affinity DataKi:  646nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265458(CHEMBL4077345)
Affinity DataKi:  660nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265508(CHEMBL4101810)
Affinity DataKi:  676nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265457(CHEMBL4083805)
Affinity DataKi:  708nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265508(CHEMBL4101810)
Affinity DataKi:  710nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265457(CHEMBL4083805)
Affinity DataKi:  720nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265456(CHEMBL4063789)
Affinity DataKi:  912nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265456(CHEMBL4063789)
Affinity DataKi:  950nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM114947(MLS001157951 | N-[2-(2-furanyl)-2-(1-pyrrolidinyl)...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM114947(MLS001157951 | N-[2-(2-furanyl)-2-(1-pyrrolidinyl)...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265506(CHEMBL4089032)
Affinity DataKi:  2.29E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265506(CHEMBL4089032)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265520(CHEMBL4099178)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265498(CHEMBL4081151)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265520(CHEMBL4099178)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265498(CHEMBL4081151)
Affinity DataKi:  2.63E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265496(CHEMBL4070528)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265497(CHEMBL4091446)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265496(CHEMBL4070528)
Affinity DataKi:  3.02E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265497(CHEMBL4091446)
Affinity DataKi:  3.02E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265519(CHEMBL4100033)
Affinity DataKi:  6.17E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265519(CHEMBL4100033)
Affinity DataKi:  6.20E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265495(CHEMBL4075479)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265495(CHEMBL4075479)
Affinity DataKi:  6.46E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265484(CHEMBL4090036)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265484(CHEMBL4090036)
Affinity DataKi:  6.61E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265526(CHEMBL4061999)
Affinity DataKi:  8.10E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50265526(CHEMBL4061999)
Affinity DataKi:  8.13E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50020493(6-Amino-5,6,7,8-tetrahydro-naphthalen-2-ol | CHEMB...)
Affinity DataKi:  8.30E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50020493(6-Amino-5,6,7,8-tetrahydro-naphthalen-2-ol | CHEMB...)
Affinity DataKi:  8.32E+3nMAssay Description:Displacement of 3H-U69593 from human KOR expressed in HEK293 cells after 90 mins by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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