Found 32 Enz. Inhib. hit(s) with all data for entry = 50000301 
Affinity DataIC50: 0.400nMAssay Description:Inhibition of rat cortex AChE using acetylthiocholine iodide as substrate measured after 8 mins in presence of BuChE inhibitor ethopropazine by Ellma...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition after 2 mins by DTN...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of BuChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of equine serum BuChE using s-butyrylthiocholine iodide as substrate pretreated for 6 mins followed by substrate addition measured at 60 s...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human plasma AChE using acetyl-(beta-methyl)thiocholine as substrate pretreated for 30 mins followed by substrate addition after 25 min...More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrateMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition after 2 mins by DTNB...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human RBC BuChE using s-butyrylthiocholine as substrate pretreated for 30 mins followed by substrate addition after 25 mins by spectrop...More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of human BuChEMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition measured at 1 min i...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate pretreated for 6 mins followed by substrate measured at 60 secs interval ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of BuChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of fetal bovine serum AChE using acetylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition by DTNB reagent b...More data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Inhibition of human plasma AChE using acetyl-(beta-methyl)thiocholine as substrate pretreated for 30 mins followed by substrate addition after 25 min...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of fetal bovine serum AChE using acetylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of human RBC BuChE using s-butyrylthiocholine as substrate pretreated for 30 mins followed by substrate addition after 25 mins by spectrop...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of recombinant human AChE expressed in HEK293 cells using acetylthiocholine chloride as substrate after 5 mins by spectrophotometric metho...More data for this Ligand-Target Pair
Affinity DataIC50: 5.71E+3nMAssay Description:Inhibition of human serum BuChE using butyrylthiocholine iodide as substrate pretreated for 20 mins followed by substrate addition by DTNB reagent ba...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition measured at 1 ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of BuChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of fetal bovine serum AChE using acetylthiocholine iodide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate measured at 12 secs interval for 10 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human plasma BuChE using butyrylthiocholine iodine as substrate pretreated for 10 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human plasma BuChE using butyrylthiocholine iodine as substrate pretreated for 10 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate measured at 12 secs interval for 10 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.60E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured at 12 secs interval for 10 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured at 12 secs interval for 10 mins by Ellman's methodMore data for this Ligand-Target Pair
