Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50049287
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 64nMAssay Description:Inhibition of human CREBBP by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238139(CHEMBL4066064)
Affinity DataIC50: 76nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238135(CHEMBL4074125)
Affinity DataIC50: 90nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50: 120nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238128(CHEMBL4101368)
Affinity DataIC50: 130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM188517(PF-CBP1)
Affinity DataIC50: 130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238153(CHEMBL4066476)
Affinity DataIC50: 130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238138(CHEMBL4093638)
Affinity DataIC50: 140nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238130(CHEMBL4063290)
Affinity DataIC50: 160nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238149(CHEMBL4074405)
Affinity DataIC50: 170nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238134(CHEMBL4085966)
Affinity DataIC50: 200nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238152(CHEMBL4075074)
Affinity DataIC50: 200nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238146(CHEMBL4103593)
Affinity DataIC50: 210nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238260(CHEMBL4094643)
Affinity DataIC50: 210nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238259(CHEMBL4096429)
Affinity DataIC50: 240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238255(CHEMBL3753333)
Affinity DataIC50: 240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238262(CHEMBL4094017)
Affinity DataIC50: 240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238151(CHEMBL4063726)
Affinity DataIC50: 260nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238136(CHEMBL4065507)
Affinity DataIC50: 300nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238258(CHEMBL4075476)
Affinity DataIC50: 310nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238142(CHEMBL4078019)
Affinity DataIC50: 310nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238263(CHEMBL4064489)
Affinity DataIC50: 330nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238146(CHEMBL4103593)
Affinity DataIC50: 350nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238261(CHEMBL4074676)
Affinity DataIC50: 360nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238131(CHEMBL4077279)
Affinity DataIC50: 400nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238254(CHEMBL4104158)
Affinity DataIC50: 400nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238140(CHEMBL4085900)
Affinity DataIC50: 450nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238256(CHEMBL4078384)
Affinity DataIC50: 470nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238139(CHEMBL4066064)
Affinity DataIC50: 490nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238148(CHEMBL4078551)
Affinity DataIC50: 500nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238145(CHEMBL4068497)
Affinity DataIC50: 500nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM188517(PF-CBP1)
Affinity DataIC50: 620nMAssay Description:Displacement of [3H]prazosin from recombinant human adrenergic A1a receptor after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238133(CHEMBL4071814)
Affinity DataIC50: 650nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238150(CHEMBL4085329)
Affinity DataIC50: 690nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238264(CHEMBL4068021)
Affinity DataIC50: 740nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238132(CHEMBL4092184)
Affinity DataIC50: 780nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238253(CHEMBL4086250)
Affinity DataIC50: 920nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238257(CHEMBL4095141)
Affinity DataIC50: 980nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238141(CHEMBL4103824)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238134(CHEMBL4085966)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238133(CHEMBL4071814)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238147(CHEMBL4076179)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238128(CHEMBL4101368)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238140(CHEMBL4085900)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238143(CHEMBL4096066)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238129(CHEMBL4084942)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238263(CHEMBL4064489)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238135(CHEMBL4074125)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238145(CHEMBL4068497)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2019
Entry Details Article
PubMed
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