Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50000650
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256930BDBM50256930(CHEMBL4097172)
Affinity DataKd:  49nMAssay Description:Binding affinity to human wild type GCK (M1 to G318 residues) expressed in mammalian expression system by KINOMEScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256917BDBM50256917(CHEMBL4084376)
Affinity DataKd:  59nMAssay Description:Binding affinity to human wild type GCK (M1 to G318 residues) expressed in mammalian expression system by KINOMEScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256918BDBM50256918(CHEMBL4088519)
Affinity DataKd:  100nMAssay Description:Binding affinity to human wild type GCK (M1 to G318 residues) expressed in mammalian expression system by KINOMEScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256919BDBM50256919(CHEMBL4103925)
Affinity DataKd:  220nMAssay Description:Binding affinity to human wild type GCK (M1 to G318 residues) expressed in mammalian expression system by KINOMEScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed