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Found 24 Enz. Inhib. hit(s) with all data for entry = 50000962
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant human C-terminal His-tagged SPHK1 expressed in fall armyworm sf21 cells using sphingosine as substrate after 1 hr by FITC-b...More data for this Ligand-Target Pair
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266429(CHEMBL4074731)
Affinity DataKi:  90nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266426(CHEMBL4076808)
Affinity DataKi:  90nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266426(CHEMBL4076808)
Affinity DataKi:  120nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266427(CHEMBL4071762)
Affinity DataKi:  170nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266428(CHEMBL4082275)
Affinity DataKi:  170nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266436(CHEMBL4093841)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266447(CHEMBL4062916)
Affinity DataKi:  300nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate by ADP-Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266425(CHEMBL4076479)
Affinity DataKi:  390nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Mus musculus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266437(CHEMBL4092871)
Affinity DataKi:  400nMAssay Description:Inhibition of recombinant mouse SPHK1 using sphingosine as substrate in presence ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266427(CHEMBL4071762)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266446(CHEMBL4074878)
Affinity DataKi:  730nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266428(CHEMBL4082275)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266425(CHEMBL4076479)
Affinity DataKi:  820nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266446(CHEMBL4074878)
Affinity DataKi:  900nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Mus musculus (Mouse))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266438(CHEMBL4095315)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of recombinant mouse SPHK2 using sphingosine as substrate in presence ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266436(CHEMBL4093841)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50017016(CHEMBL3287036)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibition of recombinant human SPHK2 at using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50312869(4-(4-(4-chlorophenyl)thiazol-2-ylamino)phenol | CH...)
Affinity DataKi:  7.90E+3nMAssay Description:Inhibition of recombinant human SPHK2 expressed in Escherichia coli using [3-3H]sphingosine as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266429(CHEMBL4074731)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate after 30 mins in presence of gamma-[32P]-ATP by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50393642(CHEMBL2158685)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of recombinant human SPHK2 using sphingosine as substrate by ADP-Quest assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266438(CHEMBL4095315)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of recombinant human SPHK1 using sphingosine as substrate in presence ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50312869(4-(4-(4-chlorophenyl)thiazol-2-ylamino)phenol | CH...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of recombinant human SPHK1 expressed in Escherichia coli using [3-3H]sphingosine as substrate after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSphingosine kinase 2(Mus musculus (Mouse))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50266437(CHEMBL4092871)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of recombinant mouse SPHK2 using sphingosine as substrate in presence ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed