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Found 11 Enz. Inhib. hit(s) with all data for entry = 50000197
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242247(CHEMBL4074268)
Affinity DataIC50:  510nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242253(CHEMBL4092304)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242254(CHEMBL4104354)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242255(CHEMBL4105000)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242256(CHEMBL4087156)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242252(CHEMBL4071511)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242251(CHEMBL4062893)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242261(CHEMBL4080120)
Affinity DataIC50:  3.23E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242246(CHEMBL4101015)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242258(CHEMBL4067399)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242260(CHEMBL4084565)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed