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Found 9 Enz. Inhib. hit(s) with all data for entry = 50048961
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50158869(CHEMBL3786182 | US10836743, Compound GSK-2879552 |...)
Affinity DataIC50:  41nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231781(CHEMBL4090528)
Affinity DataIC50:  564nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231773(CHEMBL4069511)
Affinity DataIC50:  678nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231771(CHEMBL4087193)
Affinity DataIC50:  685nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231780(CHEMBL4065771)
Affinity DataIC50:  717nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231778(CHEMBL4068480)
Affinity DataIC50:  758nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231754(CHEMBL4074390)
Affinity DataIC50:  960nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231769(CHEMBL4094875)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Technology Of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50231776(CHEMBL4095820)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed