Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50001003
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069989BDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 4nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267379BDBM50267379(CHEMBL4076340)
Affinity DataIC50: 57nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267412BDBM50267412(CHEMBL4102943)
Affinity DataIC50: 67nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267377BDBM50267377(CHEMBL4062305)
Affinity DataIC50: 75nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267378BDBM50267378(CHEMBL4084020)
Affinity DataIC50: 90nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267414BDBM50267414(CHEMBL4087490)
Affinity DataIC50: 99nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267359BDBM50267359(CHEMBL4105439)
Affinity DataIC50: 110nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267361BDBM50267361(CHEMBL4087567)
Affinity DataIC50: 168nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267388BDBM50267388(CHEMBL4076043)
Affinity DataIC50: 182nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267411BDBM50267411(CHEMBL4061779)
Affinity DataIC50: 197nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267357BDBM50267357(CHEMBL4083955)
Affinity DataIC50: 237nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267358BDBM50267358(CHEMBL4070848)
Affinity DataIC50: 740nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267364BDBM50267364(CHEMBL4103403)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267376BDBM50267376(CHEMBL4084717)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267348BDBM50267348(CHEMBL4074327)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267413BDBM50267413(CHEMBL4076234)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267349BDBM50267349(CHEMBL4105518)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267350BDBM50267350(CHEMBL4087634)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267356BDBM50267356(CHEMBL4062228)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome beta 5 subunit in human U266 cells using Suc-LLVY-aminoluciferin as substrate after 1 hr b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2020
Entry Details Article
PubMed