Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50000406
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445054BDBM50445054(CHEMBL3098745 | US9682967, 1 | US10195186, Example...)
Affinity DataIC50: 316nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249504BDBM50249504(CHEMBL4063871)
Affinity DataIC50: 3.98E+3nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249497BDBM50249497(CHEMBL4081074)
Affinity DataIC50: 1.26E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249494BDBM50249494(CHEMBL4065805)
Affinity DataIC50: 1.26E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249476BDBM50249476(CHEMBL4091656)
Affinity DataIC50: 1.26E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249487BDBM50249487(CHEMBL4098559)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249474BDBM50249474(CHEMBL4101877)
Affinity DataIC50: 3.16E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249505BDBM50249505(CHEMBL4071744)
Affinity DataIC50: 3.16E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249495BDBM50249495(CHEMBL4076922)
Affinity DataIC50: 3.98E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249473BDBM50249473(CHEMBL4068508)
Affinity DataIC50: 3.98E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249503BDBM50249503(CHEMBL4094145)
Affinity DataIC50: 5.01E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249475BDBM50249475(CHEMBL4083880)
Affinity DataIC50: 6.31E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249496BDBM50249496(CHEMBL4081301)
Affinity DataIC50: 6.31E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249499BDBM50249499(CHEMBL4100027)
Affinity DataIC50: 6.31E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249472BDBM50249472(CHEMBL4094813)
Affinity DataIC50: 7.94E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249500BDBM50249500(CHEMBL4104384)
Affinity DataIC50: 7.94E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249502BDBM50249502(CHEMBL4067376)
Affinity DataIC50: 1.26E+5nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427208BDBM50427208(CHEMBL554820)
Affinity DataIC50: 1.26E+5nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249498BDBM50249498(CHEMBL4095207)
Affinity DataIC50: 1.26E+5nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetSortilin(Human)
Aarhus University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249506BDBM50249506(CHEMBL1709220)
Affinity DataIC50: 1.58E+5nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed