Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50000527
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252472(CHEMBL4085914)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252483(CHEMBL4081524)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252452(CHEMBL4074797)
Affinity DataIC50:  6.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240170(CHEMBL4064816)
Affinity DataIC50:  9.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252462(CHEMBL4104333)
Affinity DataIC50:  9.90nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252484(CHEMBL4059569)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252509(CHEMBL4060696)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252464(CHEMBL4081022)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252510(CHEMBL4076413)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252481(CHEMBL4079088)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252494(CHEMBL4105272)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252465(CHEMBL4088913)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252492(CHEMBL4062313)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252508(CHEMBL4096603)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252480(CHEMBL4097108)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252454(CHEMBL4079668)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252453(CHEMBL4066183)
Affinity DataIC50:  60nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252479(CHEMBL4089322)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252466(CHEMBL4063118)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252475(CHEMBL4069825)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252460(CHEMBL4069371)
Affinity DataIC50:  97nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252485(CHEMBL4070938)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252473(CHEMBL4104745)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252493(CHEMBL4090320)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252497(CHEMBL4087549)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252461(CHEMBL4080094)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252457(CHEMBL4063975)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252458(CHEMBL4088446)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252498(CHEMBL4068881)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252455(CHEMBL4103920)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252512(CHEMBL4061154)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252514(CHEMBL4073810)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252482(CHEMBL4089396)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252516(CHEMBL4097566)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252515(CHEMBL4101880)
Affinity DataIC50:  470nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252496(CHEMBL4088911)
Affinity DataIC50:  750nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252463(CHEMBL4099055)
Affinity DataIC50:  2.50E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252511(CHEMBL4097022)
Affinity DataIC50:  4.20E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252474(CHEMBL4080521)
Affinity DataIC50:  4.90E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252471(CHEMBL4090279)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252459(CHEMBL4077663)
Affinity DataIC50:  7.80E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252456(CHEMBL4096167)
Affinity DataIC50:  7.90E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252517(CHEMBL4076480)
Affinity DataIC50:  7.95E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252495(CHEMBL4081019)
Affinity DataIC50:  8.70E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252499(CHEMBL4095679)
Affinity DataIC50:  8.80E+3nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed