Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50001518
TargetCruzipain(Trypanosoma cruzi)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50114613((1E)-1-(3-bromophenyl)propan-1-one thiosemicarbazo...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Trypanosoma cruzi cruzipain using Bz-Pro-Phe-Arg-p-NA as a chromogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50282195(CHEMBL4172128)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzipain using Bz-Pro-Phe-Arg-p-NA as a chromogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50282196(CHEMBL4168973)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzipain using Bz-Pro-Phe-Arg-p-NA as a chromogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50282194(CHEMBL4161560)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzipain using Bz-Pro-Phe-Arg-p-NA as a chromogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50282193(CHEMBL4176677)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzipain using Bz-Pro-Phe-Arg-p-NA as a chromogenic substrate preincubated for 10 mins followed by substrate additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed