Found 28 Enz. Inhib. hit(s) with all data for entry = 50001505 TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Histamine H2 receptor antagonistic activity at a concentration of 1 uM on the isolated guinea pig right atrium.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Histamine H2 receptor antagonistic activity at a concentration of 1 uM on the isolated guinea pig right atrium.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Reversible competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Reversible competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.75E+4nMAssay Description:Inhibition of equine serum BChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.28E+4nMAssay Description:Reversible competitive inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.62E+4nMAssay Description:Histamine H1 receptor antagonistic activity on the isolated guinea pig ileum determined by Schild plot.More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+4nMAssay Description:Inhibition of equine serum BChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+4nMAssay Description:Reversible competitive inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of human brain cortex AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
3D Structure (crystal)TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+4nMAssay Description:Histamine H1 receptor antagonistic activity on the isolated guinea pig ileum determined by Schild plot.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+4nMAssay Description:Histamine H1 receptor antagonistic activity on the isolated guinea pig ileum determined by Schild plot.More data for this Ligand-Target Pair
Affinity DataIC50: 4.94E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+5nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+5nMAssay Description:Reversible competitive inhibition of equine serum BChE using acetylthiocholine iodide as substrate measured over 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+5nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.31E+5nMAssay Description:Histamine H2 receptor antagonistic activity at a concentration of 1 uM on the isolated guinea pig right atrium.More data for this Ligand-Target Pair
