Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50000538
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252943(CHEMBL4082672)
Affinity DataEC50:  1.17E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252944(CHEMBL2046559)
Affinity DataEC50:  3.95E+3nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252945(CHEMBL4068115)
Affinity DataEC50:  3.27E+3nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252960(CHEMBL4063260)
Affinity DataEC50:  1.11E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252957(CHEMBL4085674)
Affinity DataEC50:  1.40E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252958(CHEMBL4071705)
Affinity DataEC50:  4.90E+3nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252959(CHEMBL4100347)
Affinity DataEC50:  1.20E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50252955(CHEMBL4090046)
Affinity DataEC50:  6.35E+3nMAssay Description:Antagonist activity at TLR4 (unknown origin) expressed in human AD293 cells assessed as inhibition of LPS/ATP-stimulated TLR4/NF-kB signaling pathway...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed