Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50000227
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242755(CHEMBL4101006)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242816(CHEMBL4093271)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242757(CHEMBL4090814)
Affinity DataEC50:  100nMAssay Description:Inhibition of purified HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242758(CHEMBL4085525)
Affinity DataEC50:  100nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242759(CHEMBL4063950)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242767(CHEMBL4072542)
Affinity DataEC50:  3.10E+3nMAssay Description:Inhibition of purified HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242768(CHEMBL4060580)
Affinity DataEC50:  7.90E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242769(CHEMBL4082468)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242770(CHEMBL4071981)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242772(CHEMBL4091218)
Affinity DataEC50:  200nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242781(CHEMBL4083428)
Affinity DataEC50:  40nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242782(CHEMBL4101417)
Affinity DataEC50:  31nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242783(CHEMBL4072997)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242784(CHEMBL4090191)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242785(CHEMBL4069128)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242786(CHEMBL4082347)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242792(CHEMBL4071846)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242793(CHEMBL4098841)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242794(CHEMBL4091097)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242795(CHEMBL4098957)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of purified HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242796(CHEMBL4063355)
Affinity DataEC50:  790nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242797(CHEMBL4093697)
Affinity DataEC50:  500nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242798(CHEMBL4060445)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of purified HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242814(CHEMBL4063218)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242815(CHEMBL4062882)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242756(CHEMBL4083023)
Affinity DataEC50:  80nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed