Affinity DataKi: 3.00E+3nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
Affinity DataKi: 6.40E+3nMAssay Description:Antagonist activity at open state of GluA1 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 2 mM glutamateMore data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:Antagonist activity at closed state of GluA4 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 100 uM gluta...More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
Affinity DataKi: 1.14E+4nMAssay Description:Antagonist activity at open state of GluA4 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 3 mM glutamateMore data for this Ligand-Target Pair
Affinity DataKi: 1.32E+4nMAssay Description:Antagonist activity at closed state of GluA1 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 40 to 50 uM ...More data for this Ligand-Target Pair
Affinity DataKi: 1.39E+4nMAssay Description:Antagonist activity at open state of GluA3 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 3 mM glutamateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
Affinity DataKi: 2.78E+4nMAssay Description:Antagonist activity at closed state of GluA3 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 100 uM gluta...More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
Affinity DataKi: 9.40E+4nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
Affinity DataKi: 1.64E+5nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair