Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50001026
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267948(CHEMBL4097333)
Affinity DataKi:  3.00E+3nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267953(CHEMBL199872)
Affinity DataKi:  4.00E+3nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50048389(4-(8-Methyl-9H-1,3-dioxa-6,7-diaza-cyclohepta[f]in...)
Affinity DataKi:  4.00E+3nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50048389(4-(8-Methyl-9H-1,3-dioxa-6,7-diaza-cyclohepta[f]in...)
Affinity DataKi:  5.00E+3nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  5.00E+3nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  6.40E+3nMAssay Description:Antagonist activity at open state of GluA1 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 2 mM glutamateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  7.40E+3nMAssay Description:Antagonist activity at closed state of GluA4 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 100 uM gluta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267953(CHEMBL199872)
Affinity DataKi:  9.00E+3nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  1.14E+4nMAssay Description:Antagonist activity at open state of GluA4 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 3 mM glutamateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  1.32E+4nMAssay Description:Antagonist activity at closed state of GluA1 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 40 to 50 uM ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  1.39E+4nMAssay Description:Antagonist activity at open state of GluA3 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 3 mM glutamateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267948(CHEMBL4097333)
Affinity DataKi:  1.40E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50175229(6-(4-amino-phenyl)-2,3,8,10-tetrahydro-1,4-dioxa-7...)
Affinity DataKi:  2.10E+4nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267951(CHEMBL4071408)
Affinity DataKi:  2.78E+4nMAssay Description:Antagonist activity at closed state of GluA3 (unknown origin) assessed as reduction in glutamate-induced current response in presence of 100 uM gluta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50175229(6-(4-amino-phenyl)-2,3,8,10-tetrahydro-1,4-dioxa-7...)
Affinity DataKi:  3.30E+4nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267947(CHEMBL4088629)
Affinity DataKi:  5.00E+4nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267947(CHEMBL4088629)
Affinity DataKi:  5.00E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267952(CHEMBL406937)
Affinity DataKi:  9.40E+4nMAssay Description:Antagonist activity at closed state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50267952(CHEMBL406937)
Affinity DataKi:  1.64E+5nMAssay Description:Antagonist activity at open state of GFP-tagged GluA2Qflip isoform (unknown origin) expressed in HEK293S cells assessed as reduction in glutamate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed