Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50001030
TargetCholinesterase(Horse)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 29nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267978BDBM50267978(CHEMBL4096931)
Affinity DataKi:  230nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267978BDBM50267978(CHEMBL4096931)
Affinity DataIC50: 460nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268001BDBM50268001(CHEMBL4100446)
Affinity DataKi:  570nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human erythrocyte acetylcholinesterase using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267979BDBM50267979(CHEMBL4069738)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268002BDBM50268002(CHEMBL4082432)
Affinity DataIC50: 830nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267979BDBM50267979(CHEMBL4069738)
Affinity DataIC50: 960nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267998BDBM50267998(CHEMBL4061796)
Affinity DataIC50: 980nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268001BDBM50268001(CHEMBL4100446)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267997BDBM50267997(CHEMBL4061056)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267977BDBM50267977(CHEMBL4080436)
Affinity DataKi:  1.61E+3nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130915BDBM50130915(CHEMBL1231178 | CHEBI:3122)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268000BDBM50268000(CHEMBL4065596)
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267982BDBM50267982(CHEMBL4100011)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268003BDBM50268003(CHEMBL4092718)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267977BDBM50267977(CHEMBL4080436)
Affinity DataIC50: 3.91E+3nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267981BDBM50267981(CHEMBL4089864)
Affinity DataKi:  6.51E+3nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267981BDBM50267981(CHEMBL4089864)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267971BDBM50267971(CHEMBL4093240)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268005BDBM50268005(CHEMBL4084517)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267970BDBM50267970(CHEMBL4104662)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268007BDBM50268007(CHEMBL4092260)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267983BDBM50267983(CHEMBL4090402)
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267996BDBM50267996(CHEMBL4099381)
Affinity DataIC50: 3.82E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50267980BDBM50267980(CHEMBL4089228)
Affinity DataIC50: 4.83E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268004BDBM50268004(CHEMBL4062840)
Affinity DataIC50: 5.34E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
Urals Branch of Russian Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268006BDBM50268006(CHEMBL4071464)
Affinity DataIC50: 5.86E+4nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate preincubated for 10 mins followed by substrate addition by spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed