Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50000413
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50072352(CHEMBL3409318)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249593(CHEMBL4070881)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50249592(CHEMBL4061179)
Affinity DataKi:  1.20nMAssay Description:Displacement of [35S]GTPgammaS from human recombinant CB2 receptor expressed in CHO cells after 60 min by liquid scintillation spectrometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50249595(CHEMBL4099487)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249594(CHEMBL4081467)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249595(CHEMBL4099487)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249594(CHEMBL4081467)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072352(CHEMBL3409318)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249593(CHEMBL4070881)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249585(CHEMBL3099055)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50249585(CHEMBL3099055)
Affinity DataIC50:  180nMAssay Description:Inhibition of CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249596(CHEMBL4083976)
Affinity DataEC50:  40nMAssay Description:Activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249597(CHEMBL4077214)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50249587(CHEMBL4069848)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249589(CHEMBL4101222)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249588(CHEMBL4089341)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human CB2 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249588(CHEMBL4089341)
Affinity DataEC50:  178nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249591(CHEMBL4097041)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249590(CHEMBL4083220)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human CB1 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50249587(CHEMBL4069848)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at human CB2 receptor expressed in mouse AtT-20 cells co expressing GIRK by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed