Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50000662
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0530nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257221(CHEMBL4059998)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257220(CHEMBL4075830)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257251(CHEMBL4069459)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257228(CHEMBL4077740)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257230(CHEMBL4076754)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257219(CHEMBL4059541)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257252(CHEMBL4076953)
Affinity DataKi:  0.150nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257234(CHEMBL4103607)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257232(CHEMBL4061039)
Affinity DataKi:  0.180nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257229(CHEMBL4098390)
Affinity DataKi:  0.190nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257231(CHEMBL4065973)
Affinity DataKi:  0.450nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257222(CHEMBL4075655)
Affinity DataKi:  0.560nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257227(CHEMBL4085677)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50257233(CHEMBL4077505)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed