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Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50001090
TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269276(CHEMBL4093632)
Affinity DataEC50:  1.42E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269282(CHEMBL4082823)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50274347((2E)-N-[(5R,6R)-17-(cyclopropylmethyl)-4,5-epoxy-3...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269278(CHEMBL4103819)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at human kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269279(CHEMBL4071546)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269280(CHEMBL4072327)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269281(CHEMBL4060942)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269282(CHEMBL4082823)
Affinity DataEC50:  0.0222nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269286(CHEMBL4069608)
Affinity DataEC50:  0.0799nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269287(CHEMBL4087151)
Affinity DataEC50:  4.87E+3nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269288(CHEMBL4090628)
Affinity DataEC50:  0.0494nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269289(CHEMBL4080324)
Affinity DataEC50:  0.0288nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269290(CHEMBL4098351)
Affinity DataEC50:  0.0953nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269291(CHEMBL4064781)
Affinity DataEC50:  0.0257nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269278(CHEMBL4103819)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269292(CHEMBL4066058)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269295(CHEMBL4098579)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269296(CHEMBL4099273)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269286(CHEMBL4069608)
Affinity DataEC50:  904nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269297(CHEMBL4086255)
Affinity DataEC50:  3.76E+3nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269298(CHEMBL4077552)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269279(CHEMBL4071546)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269295(CHEMBL4098579)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269296(CHEMBL4099273)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269280(CHEMBL4072327)
Affinity DataEC50:  1.29E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269287(CHEMBL4087151)
Affinity DataEC50:  0.00466nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269292(CHEMBL4066058)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269276(CHEMBL4093632)
Affinity DataEC50:  0.122nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269278(CHEMBL4103819)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269288(CHEMBL4090628)
Affinity DataEC50:  308nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269297(CHEMBL4086255)
Affinity DataEC50:  0.291nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269298(CHEMBL4077552)
Affinity DataEC50:  0.0283nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269289(CHEMBL4080324)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269290(CHEMBL4098351)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269291(CHEMBL4064781)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50269281(CHEMBL4060942)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO-dhfr(-) cells assessed as inhibition of forskolin-induced cAMP accumulation by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50274347((2E)-N-[(5R,6R)-17-(cyclopropylmethyl)-4,5-epoxy-3...)
Affinity DataEC50:  0.00820nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)