Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50002285
TargetSubstance-P receptor(Human)
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50456633(CHEMBL4215185)
Affinity DataEC50:  3.50E+5nMAssay Description:Partial agonist activity at His6-tagged NK1 receptor (unknown origin) expressed in CHO cells assessed as IP1 accumulation measured after 30 mins by H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50456631(CHEMBL4206396)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at His6-tagged NK1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of substance-P-induced IP1 accumulatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50002653(CHEMBL419500 | ((2R,3S)-2-Benzhydryl-1-aza-bicyclo...)
Affinity DataIC50: 8.10E+4nMAssay Description:Antagonist activity at His6-tagged NK1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of substance-P-induced IP1 accumulatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50456632(CHEMBL4214013)
Affinity DataIC50: 2.00E+5nMAssay Description:Antagonist activity at His6-tagged NK1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of substance-P-induced IP1 accumulatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed