Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50000777
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataKi:  1.33E+3nMAssay Description:Uncompetitive inhibition of cathepsin L (unknown origin) peincubated for 30 mins followed by substrate Z-FR-MCA addition measured after 10 mins by sp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.02E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260366(CHEMBL4065391)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human liver cathepsin L peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.13E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 5.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.26E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 6 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.72E+3nMAssay Description:Inhibition of cathepsin K (unknown origin) peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 5.75E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 8 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 6.09E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 9 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 7.17E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260367(CHEMBL4102075)
Affinity DataIC50: 8.55E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 7 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 9.78E+3nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 5 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.11E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 4.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.15E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 4 uM of substrate Z-FR-MCA measured after 10 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260365(CHEMBL4096825)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of cathepsin K (unknown origin) peincubated for 5 mins followed by Z-FR-MCA addition by spectrofluorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Federal University of S£O Carlos

Curated by ChEMBL
LigandPNGBDBM50260364(CHEMBL4065603)
Affinity DataIC50: 1.69E+4nMAssay Description:Reversible inhibition of human liver cathepsin L peincubated for 30 mins followed by addition of 3.5 uM of substrate Z-FR-MCA measured after 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2020
Entry Details Article
PubMed