Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50000682
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50261110(CHEMBL493982 | Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in TRAP-stimulated platelet aggregation preincubated for 20 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50261110(CHEMBL493982 | Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-...)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in TRAP-stimulated platelet aggregation preincubated for 20 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50261110(CHEMBL493982 | Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-...)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257953(CHEMBL4101591)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in thrombin-stimulated platelet aggregation preincubated for 3 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257953(CHEMBL4101591)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in thrombin-stimulated platelet aggregation preincubated for 3 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258055(CHEMBL4084812)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257953(CHEMBL4101591)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258008(CHEMBL4069403)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258033(CHEMBL4077763)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258034(CHEMBL4091623)
Affinity DataIC50:  8.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258011(CHEMBL4065905)
Affinity DataIC50:  8.70E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258025(CHEMBL4101239)
Affinity DataIC50:  9.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258026(CHEMBL4065873)
Affinity DataIC50:  9.50E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257976(CHEMBL4092540)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258031(CHEMBL4069486)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257975(CHEMBL4093491)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258013(CHEMBL4062114)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258021(CHEMBL4100310)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258027(CHEMBL4071756)
Affinity DataIC50:  1.90E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257983(CHEMBL4072202)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257984(CHEMBL4092965)
Affinity DataIC50:  2.10E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258017(CHEMBL4083850)
Affinity DataIC50:  2.30E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258009(CHEMBL4095795)
Affinity DataIC50:  2.90E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257972(CHEMBL4066290)
Affinity DataIC50:  3.20E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258032(CHEMBL4088070)
Affinity DataIC50:  5.50E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257971(CHEMBL4074902)
Affinity DataIC50:  8.70E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258059(CHEMBL4078212)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258058(CHEMBL4093859)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258035(CHEMBL4073470)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258029(CHEMBL4085223)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258028(CHEMBL4066363)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258024(CHEMBL4074508)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258023(CHEMBL4077889)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258022(CHEMBL4092571)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258012(CHEMBL4070740)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50258010(CHEMBL4092762)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257999(CHEMBL4104430)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257998(CHEMBL4080194)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257997(CHEMBL4096709)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257982(CHEMBL4063603)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257981(CHEMBL4074969)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257980(CHEMBL4101654)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257979(CHEMBL4093927)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257978(CHEMBL4104074)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257977(CHEMBL4086167)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257974(CHEMBL4104026)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257973(CHEMBL4086105)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257940(CHEMBL4064870)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257952(CHEMBL4102764)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed