Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50035605
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252861BDBM50252861(H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]-Thr-NH2 | CHEM...)
Affinity DataIC50: 2.80nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019567BDBM50019567(CHEMBL413950 | D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr...)
Affinity DataIC50: 3.5nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019572BDBM50019572(CHEMBL437283 | D-Phe-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr...)
Affinity DataIC50: 3.70nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50367297BDBM50367297(CHEMBL1790572)
Affinity DataIC50: 5.5nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81767BDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 6nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019575BDBM50019575(19-(2-Amino-3-phenyl-propionylamino)-10-butyl-16-(...)
Affinity DataIC50: 9.60nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019573BDBM50019573(CHEMBL384284 | D-PhGly-Cys-Tyr-D-Trp-Lys-Thr-Pen-T...)
Affinity DataIC50: 350nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019570BDBM50019570(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50: 539nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019569BDBM50019569(CHEMBL274400 | D-Phe-Cys-Tyr--Trp-Lys-Thr-Pen-Thr-...)
Affinity DataIC50: 1.35E+3nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50367297BDBM50367297(CHEMBL1790572)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81767BDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019566BDBM50019566(2-{[10-(4-Amino-butyl)-19-(2-amino-2-phenyl-acetyl...)
Affinity DataIC50: 2.10E+3nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019573BDBM50019573(CHEMBL384284 | D-PhGly-Cys-Tyr-D-Trp-Lys-Thr-Pen-T...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019567BDBM50019567(CHEMBL413950 | D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019575BDBM50019575(19-(2-Amino-3-phenyl-propionylamino)-10-butyl-16-(...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019572BDBM50019572(CHEMBL437283 | D-Phe-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019576BDBM50019576(2-{[10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-ph...)
Affinity DataIC50: 9.10E+3nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252861BDBM50252861(H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]-Thr-NH2 | CHEM...)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019576BDBM50019576(2-{[10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-ph...)
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019566BDBM50019566(2-{[10-(4-Amino-butyl)-19-(2-amino-2-phenyl-acetyl...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019570BDBM50019570(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019569BDBM50019569(CHEMBL274400 | D-Phe-Cys-Tyr--Trp-Lys-Thr-Pen-Thr-...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed