Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50000694
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258891BDBM50258891(CHEMBL4067466)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335711BDBM50335711(N-2,6-bis4-methoxyphenyl)pyrimidin-4-yl)acetamide ...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335731BDBM50335731(N-2,6-bis2,4-dimethoxyphenyl)pyrimidin-4-yl)acetam...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258884BDBM50258884(CHEMBL4097170)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258888BDBM50258888(CHEMBL4096414)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258870BDBM50258870(CHEMBL4076880)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258883BDBM50258883(CHEMBL4089461)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258869BDBM50258869(CHEMBL4099480)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258887BDBM50258887(CHEMBL4093538)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258869BDBM50258869(CHEMBL4099480)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258892BDBM50258892(CHEMBL4068284)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258891BDBM50258891(CHEMBL4067466)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258870BDBM50258870(CHEMBL4076880)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258869BDBM50258869(CHEMBL4099480)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258893BDBM50258893(CHEMBL4098099)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258889BDBM50258889(CHEMBL4088707)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258890BDBM50258890(CHEMBL4094007)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258870BDBM50258870(CHEMBL4076880)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258876BDBM50258876(CHEMBL4059638)
Affinity DataKi:  353nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in human HeLa cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258876BDBM50258876(CHEMBL4059638)
Affinity DataKi:  579nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258876BDBM50258876(CHEMBL4059638)
Affinity DataKi:  668nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258886BDBM50258886(CHEMBL4079152)
Affinity DataKi:  781nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2019
Entry Details Article
PubMed