Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50035627
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019624(CHEMBL594 | 1-(2-Ethoxy-ethyl)-2-(4-methyl-[1,4]di...)
Affinity DataIC50: 6.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019595(CHEMBL276735 | 2-(4-Methyl-piperazin-1-yl)-1-(2-ph...)
Affinity DataIC50: 6.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019605(CHEMBL275383 | 1-(2-Ethoxy-ethyl)-2-(4-pentyl-[1,4...)
Affinity DataIC50: 7.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019643(CHEMBL17795 | 2-(4-Butyl-[1,4]diazepan-1-yl)-1-(2-...)
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019644(CHEMBL416357 | 1-(2-Ethoxy-ethyl)-2-(4-propyl-[1,4...)
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019602(CHEMBL273315 | 1-(2-Ethoxy-ethyl)-2-(4-hexyl-piper...)
Affinity DataIC50: 8.60nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019628(CHEMBL418731 | 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(...)
Affinity DataIC50: 9.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019609(CHEMBL279875 | 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(...)
Affinity DataIC50: 9.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019607(CHEMBL430338 | 1-(2-Ethoxy-ethyl)-2-(4-methyl-pipe...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019636(CHEMBL18123 | 2-(4-Methyl-piperazin-1-yl)-1-(2-vin...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019618(CHEMBL18233 | 1-(2-Allyloxy-ethyl)-2-(4-methyl-[1,...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019614(CHEMBL18561 | 1-(2-Butoxy-ethyl)-2-(4-methyl-[1,4]...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019629(CHEMBL278053 | 1-(2-Ethoxy-ethyl)-2-piperazin-1-yl...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019596(CHEMBL277311 | 2-(4-Methyl-piperazin-1-yl)-1-(2-pr...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019634(CHEMBL279872 | 1-(2-Methoxy-ethyl)-2-(4-methyl-pip...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019597(CHEMBL278504 | 2-(4-Butyl-piperazin-1-yl)-1-(2-eth...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019625(CHEMBL18255 | 2-(4-Benzyl-[1,4]diazepan-1-yl)-1-(2...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019631(CHEMBL18151 | 1-(2-Ethoxy-ethyl)-2-(4-propyl-piper...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019611(CHEMBL18234 | 2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019630(CHEMBL17474 | 1-(2-Ethoxy-ethyl)-2-(4-ethyl-[1,4]d...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019617(CHEMBL17876 | 1-(2-Allyloxy-ethyl)-2-(4-methyl-pip...)
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019616(CHEMBL17246 | 1-Benzyl-2-(4-methyl-piperazin-1-yl)...)
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019635(CHEMBL18060 | 1-(2-Ethoxy-ethyl)-2-(4-ethyl-pipera...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019619(CHEMBL17349 | 2-(4-Methyl-piperazin-1-yl)-1-propox...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019593(CHEMBL17893 | 1-(2-Ethylsulfanyl-ethyl)-2-(4-methy...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019626(CHEMBL17555 | 2-(4-Methyl-piperazin-1-yl)-1-pentyl...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019599(CHEMBL273320 | 2-(4-Methyl-piperazin-1-yl)-1-(2-pr...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019639(CHEMBL274747 | 2-[1,4]Diazepan-1-yl-1-(2-ethoxy-et...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019632(CHEMBL278457 | 1-Hexyl-2-(4-methyl-piperazin-1-yl)...)
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019627(CHEMBL17742 | 2-(4-Benzyl-piperazin-1-yl)-1-(2-eth...)
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019601(CHEMBL18181 | 1-(2-Ethoxy-ethyl)-2-(4-pentyl-piper...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019592(CHEMBL280255 | 1-(2-Ethoxy-ethyl)-2-(4-phenethyl-p...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019613(CHEMBL276070 | 1-(2-Butoxy-ethyl)-2-(4-methyl-pipe...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019594(CHEMBL18122 | 2-{2-[2-(4-Methyl-piperazin-1-yl)-be...)
Affinity DataIC50: 42nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019620(CHEMBL278456 | 1-Butyl-2-(4-methyl-piperazin-1-yl)...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019633(CHEMBL276774 | 2-(4-Methyl-piperazin-1-yl)-1-propy...)
Affinity DataIC50: 68nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019598(CHEMBL17946 | 1-Heptyl-2-(4-methyl-piperazin-1-yl)...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019610(CHEMBL17763 | 2-(4-Methyl-piperazin-1-yl)-1-phenet...)
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019608(CHEMBL17959 | Ethyl-{2-[2-(4-methyl-piperazin-1-yl...)
Affinity DataIC50: 290nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019622(CHEMBL277749 | 1-Methyl-2-(4-methyl-piperazin-1-yl...)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019606(CHEMBL18062 | 2-(4-Methyl-piperazin-1-yl)-1-propyl...)
Affinity DataIC50: 380nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019641(CHEMBL277956 | 2-[2-(4-Methyl-piperazin-1-yl)-benz...)
Affinity DataIC50: 410nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019637(CHEMBL17808 | 1-(2-Benzyloxy-ethyl)-2-(4-methyl-pi...)
Affinity DataIC50: 430nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019612(CHEMBL16939 | 1-(2-Methyl-pentyl)-2-(4-methyl-pipe...)
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019603(CHEMBL17655 | 1-(3-Ethylsulfanyl-propyl)-2-(4-meth...)
Affinity DataIC50: 530nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019642(CHEMBL16938 | 2-(4-Methyl-piperazin-1-yl)-1-phenyl...)
Affinity DataIC50: 760nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019600(CHEMBL17556 | 1-(3-Methoxy-propyl)-2-(4-methyl-pip...)
Affinity DataIC50: 860nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019621(CHEMBL17635 | 1-(1-Methyl-butyl)-2-(4-methyl-piper...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50019645(CHEMBL279621 | 1-(3-Methyl-butyl)-2-(4-methyl-pipe...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
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