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Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50000827
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261349(CHEMBL4073785)
Affinity DataIC50:  2nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261349(CHEMBL4073785)
Affinity DataIC50:  2nMAssay Description:Inhibition of DNA-PK in human HeLa nuclear extracts incubated for 40 mins using calf thymus DNA and fluoroscein-p53[Ser15]-peptide by Lanthascreen ti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human DNA-PK catalytic subunit using DNA and [EPPLSQEAFADLWKK] peptide substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261337(CHEMBL4074385)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM50261355(CHEMBL4071376)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM50261354(CHEMBL4103756)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261329(CHEMBL4077367)
Affinity DataIC50:  2.75E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261339(CHEMBL4079378)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261347(CHEMBL4104565)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261350(CHEMBL4091681)
Affinity DataIC50:  2.95E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261328(CHEMBL4083912)
Affinity DataIC50:  3.01E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261351(CHEMBL4062189)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261352(CHEMBL4088661)
Affinity DataIC50:  3.07E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261329(CHEMBL4077367)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261348(CHEMBL4075473)
Affinity DataIC50:  5.68E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261340(CHEMBL4084755)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50027176(2-Acetoxy-Benzoic Acid | 3-Isobutyl-Methylxanthine...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261353(CHEMBL4061587)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261341(CHEMBL4094832)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM50261338(CHEMBL4071051)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50261330(CHEMBL4105146)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed