Compile Data Set for Download or QSAR
Report error Found 117 Enz. Inhib. hit(s) with all data for entry = 50001381
LigandChemical structure of BindingDB Monomer ID 50277401BDBM50277401(CHEMBL4168440)
Affinity DataEC50:  0.600nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277418BDBM50277418(CHEMBL4159635)
Affinity DataEC50:  1.20nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277421BDBM50277421(CHEMBL4172744)
Affinity DataEC50:  2nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444007BDBM50444007(CHEMBL3092485)
Affinity DataEC50:  3.5nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277397BDBM50277397(CHEMBL4171304)
Affinity DataEC50:  4nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277423BDBM50277423(CHEMBL4176228)
Affinity DataEC50:  4nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277393BDBM50277393(CHEMBL4160529)
Affinity DataEC50:  4nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444023BDBM50444023(CHEMBL3092486)
Affinity DataEC50:  4.70nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277404BDBM50277404(CHEMBL4161427)
Affinity DataEC50:  5nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277399BDBM50277399(CHEMBL4166863)
Affinity DataEC50:  6nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444023BDBM50444023(CHEMBL3092486)
Affinity DataEC50:  7.40nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as potentiation of mitoxantrone-induced cell growth inhibition after 72 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277393BDBM50277393(CHEMBL4160529)
Affinity DataEC50:  9.70nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as potentiation of mitoxantrone-induced cell growth inhibition after 72 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277405BDBM50277405(CHEMBL4165918)
Affinity DataEC50:  10nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277426BDBM50277426(CHEMBL4172203)
Affinity DataEC50:  11nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277400BDBM50277400(CHEMBL4176534)
Affinity DataEC50:  11nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277398BDBM50277398(CHEMBL4171781)
Affinity DataEC50:  12nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444023BDBM50444023(CHEMBL3092486)
Affinity DataEC50:  13nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as potentiation of SN-38-induced cell growth inhibition after 72 hrs by MTT ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277440BDBM50277440(CHEMBL4160887)
Affinity DataEC50:  14nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277393BDBM50277393(CHEMBL4160529)
Affinity DataEC50:  16nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as potentiation of SN-38-induced cell growth inhibition after 72 hrs by MTT ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277396BDBM50277396(CHEMBL4172857)
Affinity DataEC50:  19nMAssay Description:Activation of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277402BDBM50277402(CHEMBL4170247)
Affinity DataIC50: 20nMAssay Description:Inhibition of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444023BDBM50444023(CHEMBL3092486)
Affinity DataIC50: 44nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444023BDBM50444023(CHEMBL3092486)
Affinity DataIC50: 44nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277393BDBM50277393(CHEMBL4160529)
Affinity DataIC50: 48nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277405BDBM50277405(CHEMBL4165918)
Affinity DataIC50: 55nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277405BDBM50277405(CHEMBL4165918)
Affinity DataIC50: 56nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277399BDBM50277399(CHEMBL4166863)
Affinity DataIC50: 66nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277399BDBM50277399(CHEMBL4166863)
Affinity DataIC50: 68nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444007BDBM50444007(CHEMBL3092485)
Affinity DataIC50: 81nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444007BDBM50444007(CHEMBL3092485)
Affinity DataIC50: 83nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277391BDBM50277391(CHEMBL4161606)
Affinity DataIC50: 84nMAssay Description:Inhibition of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50305083BDBM50305083(Ko143 | Ko-143 | 3-((3S,6S)-6-Isobutyl-9-methoxy-1...)
Affinity DataIC50: 84nMAssay Description:Inhibition of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50277425BDBM50277425(CHEMBL4164537)
Affinity DataIC50: 87nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277425BDBM50277425(CHEMBL4164537)
Affinity DataIC50: 87nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277395BDBM50277395(CHEMBL4161193)
Affinity DataIC50: 89nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277401BDBM50277401(CHEMBL4168440)
Affinity DataIC50: 95nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277422BDBM50277422(CHEMBL4163316)
Affinity DataIC50: 107nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277422BDBM50277422(CHEMBL4163316)
Affinity DataIC50: 107nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277394BDBM50277394(CHEMBL4176120)
Affinity DataIC50: 108nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277429BDBM50277429(CHEMBL4169350)
Affinity DataIC50: 120nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277400BDBM50277400(CHEMBL4176534)
Affinity DataIC50: 120nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277400BDBM50277400(CHEMBL4176534)
Affinity DataIC50: 121nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277419BDBM50277419(CHEMBL4172917)
Affinity DataIC50: 127nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50033324BDBM50033324((3-Nitro-phenyl)-(2-phenyl-quinazolin-4-yl)-amine ...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277423BDBM50277423(CHEMBL4176228)
Affinity DataIC50: 135nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50444024BDBM50444024(CHEMBL3092488)
Affinity DataIC50: 136nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277423BDBM50277423(CHEMBL4176228)
Affinity DataIC50: 139nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277404BDBM50277404(CHEMBL4161427)
Affinity DataIC50: 151nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277411BDBM50277411(CHEMBL4171726)
Affinity DataIC50: 166nMAssay Description:Inhibition of human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in Hoechst 33342 efflux preincubated for 30 mins followed by Hoech...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50277428BDBM50277428(CHEMBL4169523)
Affinity DataIC50: 180nMAssay Description:Inhibition of ABCG2 ATPase activity (unknown origin) expressed in baculovirus infected high5 cell membranes after 20 mins by ascorbic acid ammonia mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
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