Compile Data Set for Download or QSAR
Report error Found 139 Enz. Inhib. hit(s) with all data for entry = 50019108
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615340BDBM50615340(CHEMBL5282076)
Affinity DataKi:  0.0620nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615347BDBM50615347(CHEMBL5277744)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615348BDBM50615348(CHEMBL5270516)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615343BDBM50615343(CHEMBL5282277)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615358BDBM50615358(CHEMBL5282803)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211957BDBM211957(US9290481, 2.5)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211958BDBM211958(US9290481, 2.6)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211955BDBM211955(US9290481, 2.3)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211956BDBM211956(US9290481, 2.4)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50076185BDBM50076185(CHEMBL3416026 | US9290481, 1.1)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211951BDBM211951(US9290481, 1.2)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211953BDBM211953(US9290481, 2.1)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211954BDBM211954(US9290481, 2.2)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 211952BDBM211952(US9290481, 1.3)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50076187BDBM50076187(CHEMBL3416027 | US9290481, 1.4)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615357BDBM50615357(CHEMBL5266861)
Affinity DataIC50: 1nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615331BDBM50615331(CHEMBL5280041)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615332BDBM50615332(CHEMBL5276953)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615329BDBM50615329(CHEMBL5268696)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615330BDBM50615330(CHEMBL5273906)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615335BDBM50615335(CHEMBL5272817)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615336BDBM50615336(CHEMBL5272260)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615333BDBM50615333(CHEMBL5266175)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615334BDBM50615334(CHEMBL5270622)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615337BDBM50615337(CHEMBL5282796)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615338BDBM50615338(CHEMBL5278972)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615315BDBM50615315(CHEMBL5275887)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615316BDBM50615316(CHEMBL5272249)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615314BDBM50615314(CHEMBL5270667)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615319BDBM50615319(CHEMBL5282393)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615320BDBM50615320(CHEMBL5281109)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615317BDBM50615317(CHEMBL5271126)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221562BDBM50221562(US8481536, 540 | CHEMBL398279 | 4-(7-(2-bromo-5-hy...)
Affinity DataKi:  1nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615318BDBM50615318(CHEMBL5269901)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615323BDBM50615323(CHEMBL5270834)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615324BDBM50615324(CHEMBL5274905)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615321BDBM50615321(CHEMBL5288239)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615322BDBM50615322(CHEMBL5287305)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615327BDBM50615327(CHEMBL5282609)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615328BDBM50615328(CHEMBL5289952)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615325BDBM50615325(CHEMBL5285217)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615326BDBM50615326(CHEMBL5278557)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615347BDBM50615347(CHEMBL5277744)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to Abl-T315I mutant (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221549BDBM50221549(CHEMBL250821 | US8481536, 547 | 4-(7-(6-chloro-2-f...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615339BDBM50615339(CHEMBL5282737)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615342BDBM50615342(CHEMBL5286051)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615352BDBM50615352(CHEMBL5266023)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 311561BDBM311561(US10155765, Example 59 | 2-[(2- aminoethyl)amino]-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615341BDBM50615341(CHEMBL5269803)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615349BDBM50615349(CHEMBL5272285)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to Abl (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
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